Collect. Czech. Chem. Commun. 1987, 52, 2758-2774
https://doi.org/10.1135/cccc19872758

Potential antihistamine agents: 4-(6,11-Dihydrodibenzo[b,e]thiepin-11-ylidene)-1-methyltetrahydrothiopyranium iodide and similar sulfonium salts derived from related tricyclic systems

Zdeněk Polívkaa, Jiří Holubeka, Miloš Buděšínskýb, Oluše Matoušováa, Emil Sváteka, Jan Metyša and Miroslav Protivaa

a Research Institute for Pharmacy and Biochemistry, 130 60 Prague 3
b Institute of Organic Chemistry and Biochemistry, Czechoslovak Academy of Sciences, 166 10 Prague 6

Individual author index pages


Other CCCC articles of these authors

  • Martina Pressová, Miloš Buděšínský and Ivan Rosenberg
    Spontaneous oligomerization of imidazolidate of 5'-O-phosphonomethyladenosine
    Symposium Series 1999, Vol. 2, pp. 281–282 [Abstract]
    Published online 2016-05-08 23:32:45
  • Jana Zachová, Ivana Císařová, Miloš Buděšínský, Radek Liboska, Zdeněk Točík and Ivan Rosenberg
    Crystal and solution structure of 5'-O-(guanosine-2'-O-phosphonomethyl)cytidine, an isopolar nonisosteric phosphonate analog of GpC
    Symposium Series 1999, Vol. 2, pp. 233–236 [Abstract]
    Published online 2016-05-08 23:30:57
  • Šárka Králíková, Miloš Buděšínský, Milena Masojídková, Ivana Kavenová and Ivan Rosenberg
    Synthesis of α-hydroxyphosphonate analogs of ApA and UV spectroscopy study on their complexes with poly(U)
    Symposium Series 1999, Vol. 2, pp. 89–91 [Abstract]
    Published online 2016-05-08 20:41:40
  • Jan Mařík, Miloš Buděšínský, Jiřina Slaninová and Jan Hlaváček
    Biologically inactive methylene-oxy analogs of oxytocin and vasopressin
    Symposium Series 2001, Vol. 4, pp. 26–27 [Abstract]
    Published online 2016-04-21 09:02:59
  • Václav Vaněk, Miloš Buděšínský, Ivana Kavenová, Markéta Rinnová and Ivan Rosenberg
    Isosteric phosphonate-pyrrolidine-based dinucleoside monophosphate analogues
    Symposium Series 2002, Vol. 5, pp. 391–392 [Abstract]
    Published online 2016-01-25 20:52:06
  • Martina Pressová, Radek Liboska, Miloš Buděšínský, Šárka Králíková, Ivana Kavenová and Ivan Rosenberg
    Oligomerisation aiming at phosphonate analogues of oligoadenylates
    Symposium Series 2002, Vol. 5, pp. 383–384 [Abstract]
    Published online 2016-01-25 20:51:50
  • Ondřej Páv, Miloš Buděšínský and Ivan Rosenberg
    2'-5' Oligoadenylate analogues with C-phosphonate internucleotide linkage
    Symposium Series 2002, Vol. 5, pp. 379–380 [Abstract]
    Published online 2016-01-25 20:51:40
  • Radek Liboska, Miloš Buděšínský, Ivana Kavenová, Ondřej Páv and Ivan Rosenberg
    Hybridization properties of 4'-branched oligonucleotides
    Symposium Series 2002, Vol. 5, pp. 365–366 [Abstract]
    Published online 2016-01-25 20:51:12
  • Marcela Krečmerová, Miloš Buděšínský and Antonín Holý
    Synthesis of optically pure N6-alkyl derivatives of (2R)-3-(adenin-9-yl)-2-hydroxypropanoic acid and related compounds
    Symposium Series 2002, Vol. 5, pp. 358–360 [Abstract]
    Published online 2016-01-25 20:50:59
  • Šárka Králíková, Miloš Buděšínský, Ivana Kavenová and Ivan Rosenberg
    α-Hydroxyphosphonate oligonucleotides: A striking DNA type?
    Symposium Series 2002, Vol. 5, pp. 356–357 [Abstract]
    Published online 2016-01-25 20:50:54
  • Zdeněk Točík, Radek Liboska, Ivan Barvík, Jr., Miloš Buděšínský, Milena Masojídková, Ivana Kavenová and Ivan Rosenberg
    Isosteric phosphonate mono- and oligonucleotides originating from 4',5'-didehydronucleoside precursors: Some synthetic possibilities and limitations
    Symposium Series 2002, Vol. 5, pp. 208–214 [Abstract]
    Published online 2016-01-25 20:40:13
  • Václav Vaněk, Miloš Buděšínský and Ivan Rosenberg
    The synthesis of monomers for prolinol-based oligonucleotides
    Symposium Series 2005, Vol. 7, pp. 483–484 [Abstract]
    Published online 2015-11-08 11:58:51
  • Zdeněk Točík, Ivan Barvík, Jr., Miloš Buděšínský and Ivan Rosenberg
    Isosteric phosphonate 3'-O-P-CH2-O-4'C internucleotide linkage: Attempts to get more data on its stereochemistry
    Symposium Series 2005, Vol. 7, pp. 481–482 [Abstract]
    Published online 2015-11-08 11:58:47
  • Šárka Králíková, Miloš Buděšínský, Radek Liboska, Ondřej Páv and Ivan Rosenberg
    2',5'-Linked oligo-3'-deoxynucleotide chimeras with chiral α-hydroxyphosphonate internucleotide linkage: Improvement of hybridisation selectivity toward RNA?
    Symposium Series 2005, Vol. 7, pp. 421–422 [Abstract]
    Published online 2015-11-08 11:57:07
  • Petr Kočalka, Markéta Rinnová, Václav Vaněk, Dominik Rejman, Ivan Votruba, Ivana Tomečková, Šárka Králíková, Magdalena Petrová, Ondřej Páv, Radek Pohl, Miloš Buděšínský, Radek Liboska, Zdeněk Točík and Ivan Rosenberg
    Novel nucleoside phosphonic acids-based inhibitors of thymidine phosphorylase
    Symposium Series 2005, Vol. 7, pp. 415–416 [Abstract]
    Published online 2015-11-08 11:56:57
  • Ivan Rosenberg, Ivan Barvik, Miloš Buděšínský, Petr Kočalka, Šárka Králíková, Radek Liboska, Ondřej Pačes, Ondřej Páv, Magdalena Petrová, Radek Pohl, Martina Pressová, Dominik Rejman, Ivan Votruba and Zdeněk Točík
    Nucleoside phosphonic acids and related oligonucleotides: Structural diversity vs biological properties
    Symposium Series 2005, Vol. 7, pp. 153–157 [Abstract]
    Published online 2015-11-08 11:51:38
  • Jiří Jiráček, Michaela Collinsová, Ivan Rosenberg, Hana Netušilová, Miloš Buděšínský and Timothy A. Garrow
    New inhibitors of human betaine-homocysteine S-methyltransferase
    Symposium Series 2005, Vol. 8, pp. 33–35 [Abstract]
    Published online 2015-11-06 12:02:21
  • David Sýkora, Lenka Žáková and Miloš Buděšínský
    Monitoring of peptide bond conformation in N-methylated peptides by RP-HPLC and NMR
    Symposium Series 2005, Vol. 8, pp. 91–93 [Abstract]
    Published online 2015-11-06 11:59:58
  • Radek Pohl, Miloš Buděšínský, Dominik Rejman, Petr Kočalka and Ivan Rosenberg
    Conformation of pyrrolidine ring in pyrrolidine nucleotide analogues
    Symposium Series 2008, Vol. 10, pp. 435–436 [Abstract]
    Published online 2015-10-30 18:44:27
  • Lenka Monincová, Jiřina Slaninová, Zdeněk Voburka, Oldřich Hovorka, Vladimír Fučík, Lenka Borovičková, Lucie Bednárová, Miloš Buděšínský, Jakub Straka and Václav Čeřovský
    Novel biologically active peptides from the venom of the solitary bee Macropis fulvipes (hymenoptera: melittidae)
    Symposium Series 2009, Vol. 11, pp. 77–80 [Abstract]
    Published online 2015-08-26 09:42:11
  • Magdalena Petrová, Miloš Buděšínský, Blanka Klepetářová and Ivan Rosenberg
    Synthesis and structural assignment of novel 5'-epimeric 3'-deoxy-3',4'-didehydronucleoside-5'-C-phosphonates
    Symposium Series 2011, Vol. 12, pp. 430–432 [Abstract]
    Published online 2015-08-20 10:23:23
  • Ondřej Šimák, Petr Pachl, Tomáš Jandušík, Jiří Brynda, Miloš Buděšínský and Ivan Rosenberg
    Bi-substrate inhibitors of human pyrimidine 5’-nucleotidases
    Symposium Series 2014, Vol. 14, pp. 381–382 [Abstract]
    Published online 2015-07-06 23:09:12
  • Magdalena Petrová, Miloš Buděšínský, Eva Zborníková, Natalia Panova, Pavel Novák and Ivan Rosenberg
    Activation of human RNase L by 5’-C-phosphonate-modified oligoadenylates
    Symposium Series 2014, Vol. 14, pp. 348–349 [Abstract]
    Published online 2015-07-06 23:07:50
  • Ondřej Páv, Eva Zborníková, Miloš Buděšínský and Ivan Rosenberg
    Phosphanucleosides containing 1-hydroxymethylphospholane 1-oxide ring
    Symposium Series 2014, Vol. 14, pp. 344–345 [Abstract]
    Published online 2015-07-06 23:07:39
  • Ondřej Kostov, Eva Zborníková, Miloš Buděšínský, Pavel Novák and Ivan Rosenberg
    Sulfur-containing phosphonate monomers for oligonucleotide synthesis
    Symposium Series 2014, Vol. 14, pp. 308–309 [Abstract]
    Published online 2015-07-06 23:06:12
  • Ivana Poláková, Miloš Buděšínský, Zdeněk Točík and Ivan Rosenberg*
    Tetrofuranose nucleoside phosphonic acids: Synthesis and properties
    2011, Vol. 76, Issue 5, pp. 503–536 [Abstract]
  • Jan Šmidrkal, Juraj Harmatha*, Miloš Buděšínský, Karel Vokáč, Zdeněk Zídek, Eva Kmoníčková, Roman Merkl and Vladimír Filip
    Modified approach for preparing (E)-stilbenes related to resveratrol, and evaluation of their potential immunobiological effects
    2010, Vol. 75, Issue 2, pp. 175–186 [Abstract]
  • Juraj Harmatha*, Miloš Buděšínský, Karel Vokáč, Milan Pavlík, Karel Grüner and Věra Laudová
    Lignan Glucosides and Serotonin Phenylpropanoids from the Seeds of Leuzea carthamoides
    2007, Vol. 72, Issue 3, pp. 334–346 [Abstract]
  • Martina Džoganová, Miloslav Černý, Miloš Buděšínský*, Martin Dračínský and Tomáš Trnka
    Epoxide Migration and Pseudo-Epoxide Migration of 1,6:2,3- and 1,6:3,4-Dianhydro-β-D-hexopyranoses. Synthesis of Some Deoxy Halo Derivatives of 1,6-Anhydro-β-D-hexopyranoses
    2006, Vol. 71, Issue 10, pp. 1497–1515 [Abstract]
  • Juraj Harmatha*, Miloš Buděšínský, Karel Vokáč, Laurence Dinan and René Lafont
    Dimeric Ecdysteroid Analogues and Their Interaction with the Drosophila Ecdysteroid Receptor
    2006, Vol. 71, Issue 8, pp. 1229–1238 [Abstract]
  • Martin Dračínský, Simona Hybelbauerová, Jan Sejbal and Miloš Buděšínský*
    Preparation and Conformational Study of B-Ring Substituted Lupane Derivatives
    2006, Vol. 71, Issue 8, pp. 1131–1160 [Abstract]
  • Martin Dračínský, Václav Richtr, Václav Křeček, Jan Sejbal, Jiří Klinot and Miloš Buděšínský*
    Preparation and Conformational Study of 19β,28-Epoxy-18α-olean-5-ene Derivatives
    2006, Vol. 71, Issue 3, pp. 387–410 [Abstract]
  • Miloš Buděšínský*, Jana Poláková, Michaela Hamerníková, Ivana Císařová, Tomáš Trnka and Miloslav Černý
    1,6-Anhydro-1-thio-β-D-glucopyranose (Thiolevoglucosan) and the Corresponding Sulfoxides and Sulfone
    2006, Vol. 71, Issue 3, pp. 311–336 [Abstract]
  • Tomáš Trtek, Miloslav Černý, Miloš Buděšínský*, Tomáš Trnka and Ivana Císařová
    Synthesis of 1,6-Anhydro-β-D-hexopyranoses Fused to the Piperidine Ring
    2005, Vol. 70, Issue 9, pp. 1429–1446 [Abstract]
  • Miloš Buděšínský, Jan Fajkoš, Jaroslav Günter and Alexander Kasal*
    Synthesis, Reactions, Conformation Analysis, and NMR Spectra of 5,10-Epoxy-5ξ,10ξ-estrane-3,17-diones
    2005, Vol. 70, Issue 4, pp. 507–518 [Abstract]
  • Tomáš Trtek, Miloslav Černý, Miloš Buděšínský*, Tomáš Trnka and Ivana Císařová
    New Heterocyclic Derivatives of 2-Amino-1,6-anhydro-2-deoxy-β-D-glucopyranose Containing 1,4-Oxazepane or Azepane Ring
    2005, Vol. 70, Issue 4, pp. 466–478 [Abstract]
  • Jindřich Karban*, Miloš Buděšínský and Jiří Kroutil
    Synthesis of 1,6-Anhydro-2,3,4-trideoxy-2,3-epimino- and 1,6-Anhydro-2,3,4-trideoxy-3,4-epimino-β-D-hexopyranoses and Their NMR and Infrared Spectra
    2004, Vol. 69, Issue 10, pp. 1939–1954 [Abstract]
  • Tomáš Trtek, Miloslav Černý, Tomáš Trnka, Miloš Buděšínský* and Ivana Císařová
    Synthesis of Some 1,4-Oxazepanes Fused with 1,6-Anhydro-β-D-hexopyranoses. 3,11,13-Trioxa-7-azatricyclo[8.2.1.02,8]tridecane Derivatives
    2004, Vol. 69, Issue 9, pp. 1818–1828 [Abstract]
  • Miroslav Šíša, Miloš Buděšínský and Ladislav Kohout*
    Synthesis and Biological Activity of 7a-Homo- and 7a,7b-Dihomo-5α-cholestane Analogues of Brassinolide
    2003, Vol. 68, Issue 11, pp. 2171–2189 [Abstract]
  • Tomáš Trtek*, Miloslav Černý, Tomáš Trnka, Miloš Buděšínský and Ivana Císařová
    Synthesis of Tricycles Based on 1,6-Anhydro-β-D-hexopyranoses Fused with Morpholine. 3,10,12-Trioxa-6-azatricyclo[7.2.1.02,7]dodecanes
    2003, Vol. 68, Issue 7, pp. 1295–1308 [Abstract]
  • Marcela Krečmerová*, Miloš Buděšínský, Milena Masojídková and Antonín Holý
    Synthesis of Optically Active N6-Alkyl Derivatives of (R)-3-(Adenin-9-yl)-2-hydroxypropanoic Acid and Related Compounds
    2003, Vol. 68, Issue 5, pp. 931–950 [Abstract]
  • Simona Koščová, Miloš Buděšínský and Jana Hodačová*
    A Facile Synthesis of Selectively Protected Linear Oligoamines
    2003, Vol. 68, Issue 4, pp. 744–750 [Abstract]
  • Jiří Kroutil*, Jindřich Karban, Tomáš Trnka, Miloš Buděšínský and Miloslav Černý
    Preparation of O-, S- and N-Benzyl Derivatives of 1,6-Anhydro-β-D-hexopyranoses via Aziridine Ring Opening
    2002, Vol. 67, Issue 12, pp. 1805–1819 [Abstract]
  • Miroslav Reschel, Miloš Buděšínský, Ivan Černý, Vladimír Pouzar and Pavel Drašar*
    Synthesis of Linear Steroid Oligoesters Based on Etienic Acid
    2002, Vol. 67, Issue 11, pp. 1709–1718 [Abstract]
  • Jan Mařík, Miloš Buděšínský, Jiřina Slaninová and Jan Hlaváček*
    Synthesis, Bioassay and NMR Study of Methyleneoxy Isosters of Oxytocin and Vasopressin
    2002, Vol. 67, Issue 3, pp. 373–392 [Abstract]
  • Karel Vokáč, Miloš Buděšínský and Juraj Harmatha*
    Minor Ecdysteroid Components of Leuzea carthamoides
    2002, Vol. 67, Issue 1, pp. 124–139 [Abstract]
  • Hana Chodounská, Miloš Buděšínský, Romana Šídová, Miroslav Šíša, Alexander Kasal and Ladislav Kohout*
    Simple NMR Determination of 5α/5β Configuration of 3-Oxosteroids
    2001, Vol. 66, Issue 10, pp. 1529–1544 [Abstract]
  • Ivan Černý*, Miloš Buděšínský, Vladimír Pouzar and Pavel Drašar
    Linear Chaining of Etienic Acid Derivatives with the Amide Bond. Synthesis of Oligomeric Steroids
    2001, Vol. 66, Issue 6, pp. 933–946 [Abstract]
  • Jindřich Karban*, Miloš Buděšínský, Miloslav Černý and Tomáš Trnka
    Synthesis and NMR Spectra of 1,6-Anhydro-2,3-dideoxy-2,3-epimino- and 1,6-Anhydro-3,4-dideoxy-3,4-epimino-β-D-hexopyranoses
    2001, Vol. 66, Issue 5, pp. 799–819 [Abstract]
  • Petr Alexander*, Antonín Holý, Miloš Buděšínský and Milena Masojídková
    Synthesis of Acyclic Nucleotide Analogues Derived from N3-Substituted Isoguanine
    2000, Vol. 65, Issue 11, pp. 1713–1725 [Abstract]
  • Ivan Černý*, Vladimír Pouzar, Miloš Buděšínský and Pavel Drašar
    Synthesis of Symmetrical Bis-Steroid Pyrazines Connected via D-Rings
    2000, Vol. 65, Issue 10, pp. 1597–1608 [Abstract]
  • Jan Hlaváček*, Renáta Marcová, Miloš Buděšínský and Jiřina Slaninová
    1-Deamino-1(15)-carba and -Dicarba Analogues of Endothelin-1
    2000, Vol. 65, Issue 3, pp. 407–424 [Abstract]
  • Martin Chadim, Miloš Buděšínský, Jana Hodačová and Jiří Závada*
    A Covalently Bound Template in the Regioselective Synthesis of Bis(tetraazacrown)s
    2000, Vol. 65, Issue 1, pp. 99–105 [Abstract]
  • Alexander Kasal*, Miloš Buděšínský, Jan Pelnař, Michael A. Bruck* and Michael F. Brown
    Structures and Synthesis of 4a-Homo-7,19-dinorsteroids, X-Ray Crystallography and NMR Spectroscopy
    1999, Vol. 64, Issue 12, pp. 2019–2034 [Abstract]
  • Barbora Slavíková, Alexander Kasal* and Miloš Buděšínský
    Autoxidation vs Hydrolysis in 16α-Acyloxy Steroids
    1999, Vol. 64, Issue 7, pp. 1125–1134 [Abstract]
  • Antonín Holý*, Miloš Buděšínský, Jaroslav Podlaha and Ivana Císařová
    Synthesis of Quaternary 1-[2-(Phosphonomethoxy)ethyl] Derivatives of 2,4-Diaminopyrimidine and Related Acyclic Nucleotide Analogs
    1999, Vol. 64, Issue 2, pp. 242–256 [Abstract]
  • Alexander Kasal, Jiří Polman and Miloš Buděšínský
    Hydrogenation of a Tetrasubstituted Double Bond: Synthesis of 5-Methyl-19-nor-5β-pregnanes
    1998, Vol. 63, Issue 10, pp. 1549–1563 [Abstract]
  • Jiří Kroutil, Tomáš Trnka, Miloš Buděšínský and Miloslav Černý
    Preparation of 2,3-Dideoxy-2,3-epimino and 3,4-Dideoxy-3,4-epimino Derivatives of 1,6-Anhydro-β-D-hexopyranoses by Mitsunobu Reaction
    1998, Vol. 63, Issue 6, pp. 813–825 [Abstract]
  • Tomáš Kraus, Miloš Buděšínský and Jiří Závada
    Novel Amphiphilic Cyclodextrins: Per[6-deoxy-6-(4,5-dicarboxy-1,2,3-triazol-1-yl)-2,3-di-O-methyl] Derivatives
    1998, Vol. 63, Issue 4, pp. 534–540 [Abstract]
  • Jaroslav Litera, Miloš Buděšínský, Ján Urban and Milan Souček
    Peptide Inhibitors of Aspartic Proteinases with Hydroxyethylene Isostere Replacement of Peptide Bond. I. Preparation of Four Diastereoisomeric (2R or 2S,4R or 4S,5S)-2-Benzyl-5-[(tert-butoxycarbonyl)amino]-4-hydroxy-6-phenylhexanoic Acids
    1998, Vol. 63, Issue 2, pp. 231–244 [Abstract]
  • Miloš Tichý, Luděk Ridvan, Miloš Buděšínský, Jiří Závada, Jaroslav Podlaha and Ivana Císařová
    Axially Chiral Bis(α-amino Acid)s and Their Deamino Analogues. Synthesis and Configurational Assignment
    1998, Vol. 63, Issue 2, pp. 211–221 [Abstract]
  • Mária Haladová, Eva Eisenreichová, Pavel Mučaji, Miloš Buděšínský and Karel Ubik
    Steroidal Saponins from Lilium candidum L.
    1998, Vol. 63, Issue 2, pp. 205–210 [Abstract]
  • Jan Sejbal, Jiří Klinot, Miloš Buděšínský and Jiří Protiva
    Functionalization of Lupane-3β,28-diyl Diacetate with Chromium(VI) Oxide. Part 2
    1997, Vol. 62, Issue 12, pp. 1905–1918 [Abstract]
  • Eva Klinotová, Václav Křeček, Jiří Klinot, Magdalena Endová, Jana Eisenreichová, Miloš Buděšínský and Martin Štícha
    Glycosylation of Triterpene Alcohols and Acids of the Lupane and A-Secolupane Series
    1997, Vol. 62, Issue 11, pp. 1776–1798 [Abstract]
  • Alexander Kasal, Barbora Slavíková, Ladislav Kohout and Miloš Buděšínský
    The Synthesis of A-Homo-B-norandrostanes: The Effect of a Hydroxyl on the Course of Hydrogenation of the ∆9-Double Bond
    1997, Vol. 62, Issue 10, pp. 1631–1641 [Abstract]
  • Hubert Hřebabecký, Miloš Buděšínský, Milena Masojídková, Zdeněk Havlas and Antonín Holý
    1-(3,5-O-Alkylidene-2-deoxy-4-C-hydroxymethyl-α-L-threo-pentofuranosyl)uracils
    1997, Vol. 62, Issue 6, pp. 957–970 [Abstract]
  • Barbora Slavíková, Alexander Kasal and Miloš Buděšínský
    Dihydrotestosterone with an Ammonium Centre in the Position 16β
    1997, Vol. 62, Issue 4, pp. 656–664 [Abstract]
  • Miroslav Kuchař, Marie Poppová, Antonín Jandera, Vladimíra Panajotovová, Hana Zůnová, Miloš Buděšínský, Hana Tomková, Alexandr Jegorov and Jan Taimr
    Chiral Forms of 4-(2',4'-Difluorobiphenyl-4-yl)-2-methyl-4-oxobutanoic Acid (Flobufen) and Its Metabolite.Synthesis and Basic Biological Properties
    1997, Vol. 62, Issue 3, pp. 498–509 [Abstract]
  • Thi Thu Huong Nguyen, Jiří Protiva, Eva Klinotová, Jiří Urban and Miroslav Protiva
    Synthesis of 24-(Piperidin-1-yl, Morpholin-4-yl and 4-Methylpiperazin-1-yl)-5β-cholan-3α-ols and Four Hydroxylated 23-(4,5-Dihydroimidazol-2-yl)-24-nor-5β-cholanes
    1997, Vol. 62, Issue 3, pp. 471–478 [Abstract]
  • Pavel Mučaji, Mária Haladová, Eva Eisenreichová, Miloš Buděšínský and Karel Ubik
    Jatropham 5-O-β-D-Glucopyranoside from Lilium candidum L.
    1996, Vol. 61, Issue 11, pp. 1662–1664 [Abstract]
  • Miloslav Černý, Tomáš Trnka and Miloš Buděšínský
    Preparation and Reactions of 2-Chloroethyl 1-Thio-β-D-glycopyranosides Derived from D-Galactose, D-Glucose, and 2-Acetamido-2-deoxy-D-glucose
    1996, Vol. 61, Issue 10, pp. 1489–1500 [Abstract]
  • Jan Sejbal, Jiří Klinot and Miloš Buděšínský
    Functionalization of Lupane with Chromium(VI) Oxide. A Remark on the Structure of Clerodone
    1996, Vol. 61, Issue 9, pp. 1371–1379 [Abstract]
  • Jan Sejbal, Jiří Klinot and Miloš Buděšínský
    Oleanane Triterpenoids Functionalized at C-25 and C-26
    1996, Vol. 61, Issue 9, pp. 1360–1370 [Abstract]
  • Alexandra Šilhánková, Karel Šindelář, Karel Dobrovský, Ivan Krejčí, Jarmila Hodková and Zdeněk Polívka
    Synthesis of New L-Proline Amides with Anticonvulsive Effect
    1996, Vol. 61, Issue 7, pp. 1085–1092 [Abstract]
  • Vladimír Valenta, Karel Dobrovský, Ivan Krejčí and Zdeněk Polívka
    Potential Antagonists of Excitatory Amino Acids and Anticonvulsants: Some Heterocyclic (±)-Pyrrolidine-2-carboxamides
    1996, Vol. 61, Issue 7, pp. 1077–1084 [Abstract]
  • Wim F. Vranken, Miloš Buděšínský, Franky Fant, Kris Boulez, Hélène Gras-Masse and Frans A. M. Borremans
    Conformational Features of a Synthetic Cyclic Peptide Corresponding to the Complete V3 Loop of the ELI HIV-1 Strain in Water
    1996, Vol. 61, Issue 5, pp. 742–750 [Abstract]
  • Alexander Kasal and Miloš Buděšínský
    Partial Modifications of Hydroxy Groups in 5-Methyl-5β-estr-9-ene Derivatives
    1996, Vol. 61, Issue 2, pp. 276–287 [Abstract]
  • Václav Suchý, Miloš Buděšínský, Karel Ubik, Daniel Grančai and Vlasta Földešiová
    NMR Determination of the Structure of Peracetylated Icariside B2 from Veratrum Lobelianum BERNH.
    1995, Vol. 60, Issue 8, pp. 1380–1385 [Abstract]
  • Dalibor Štys, Ján Novák, Viktor Krchňák, Josef Vágner, Petr Štrop and Miloš Buděšínský
    Time Dependence of Immunoresponse of Different Epitopes of gp41 and Its Relation to the Structure of Short Peptide Fragments of gp41
    1995, Vol. 60, Issue 6, pp. 1054–1064 [Abstract]
  • Karel Šindelář, Karel Dobrovský, Ivan Krejčí and Zdeněk Polívka
    Substituted 1-(2-Thienyl)cyclohexylamines and Related Compounds as Potential NMDA Antagonists
    1995, Vol. 60, Issue 5, pp. 894–902 [Abstract]
  • Václav Křeček, Stanislav Hilgard, Miloš Buděšínský and Alois Vystrčil
    E-Homolupane Derivatives Substituted in Position 17 and 22a. 1H NMR, 13C NMR and IR Spectra
    1995, Vol. 60, Issue 4, pp. 619–635 [Abstract]
  • Miloš Buděšínský, Miloslav Černý, Ivan Černý, Stanislav Sámek and Tomáš Trnka
    Preparation of β-D-Glucopyranosyl Derivatives of 1,6:2,3- and 1,6:3,4-Dianhydro-β-D-hexopyranoses and Their 1H and 13C NMR Spectra
    1995, Vol. 60, Issue 2, pp. 311–323 [Abstract]
  • Urszula Rychłewska, Miloš Buděšínský, Halina Grabarczyk, Bohdan Drożdż and Miroslav Holub
    X-Ray Structure Analysis and NMR Study of Sesquiterpene Lactone Hirsutolide
    1995, Vol. 60, Issue 2, pp. 300–310 [Abstract]
  • Urszula Rychłewska, Miloš Buděšínský, Beata Szczepanska, Ełżbieta Błoszyk and Miroslav Holub
    Two Crystalline Forms of Sesquiterpene Lactone Helenalin - X-Ray and NMR Study
    1995, Vol. 60, Issue 2, pp. 276–299 [Abstract]
  • Thi Thu Huong Nguyen, Jiří Urban, Eva Klinotová, Jan Sejbal, Jiří Protiva, Pavel Drašar and Miroslav Protiva
    Synthesis of Several Hydroxylated 23-(Benzimidazol-2-yl-, Benzoxazol-2-yl and Benzothiazol-2-yl)norcholanes and Some Related Compounds
    1995, Vol. 60, Issue 2, pp. 257–275 [Abstract]
  • Dana Hocková, Milena Masojídková, Miloš Buděšínský and Antonín Holý
    Acyclic Nucleoside and Nucleotide Analogs Derived from 2-Azaadenine
    1995, Vol. 60, Issue 2, pp. 224–236 [Abstract]
  • Ivan Černý, Miloš Buděšínský, Pavel Drašar and Vladimír Pouzar
    Construction of the Side-Chain in 14β-Androst-5-ene Derivatives. Preparation of 14β-Pregnenolone
    1994, Vol. 59, Issue 12, pp. 2691–2704 [Abstract]
  • Vojtěch Kmoníček, Martin Valchář and Zdeněk Polívka
    Some 4-Substituted 1-(3-Pyridylmethyl)piperazines with Antihistamine Activity
    1994, Vol. 59, Issue 10, pp. 2343–2350 [Abstract]
  • Miloš Buděšínský, Gerard Nowak, Urszula Rychłewska, Derek J. Hodgson, David Šaman, Włodzimierz M. Daniewski, Bohdan Drożdż and Miroslav Holub
    Structure of Sesquiterpenic Lactones of Some Species of Subtribe Centaureinae DUMORT.
    1994, Vol. 59, Issue 5, pp. 1175–1202 [Abstract]
  • Maria Spassova, Hana Dvořáková, Antonín Holý, Miloš Buděšínský and Milena Masojídková
    Synthesis of N-(3-Azido-2-hydroxypropyl), N-(3-Phthalimido-2-hydroxypropyl) and N-(3-Amino-2-hydroxypropyl) Derivatives of Heterocyclic Bases
    1994, Vol. 59, Issue 5, pp. 1153–1174 [Abstract]
  • Vladimír Valenta, Jiří Urban, Jan Taimr and Zdeněk Polívka
    Potential Nootropic Agents: Synthesis of Some 1,4-Disubstituted 2-Oxopyrrolidines and Some Related Compounds
    1994, Vol. 59, Issue 5, pp. 1126–1136 [Abstract]
  • Miloš Buděšínský, Nestor Perez Souto and Miroslav Holub
    Sesquiterpenic Lactones of Some Species of Genus Vernonia SCHREB.
    1994, Vol. 59, Issue 4, pp. 913–928 [Abstract]
  • Karel Šindelář, Alexandra Šilhánková, Jiří Urban, Jan Metyš, Martin Valchář and Zdeněk Polívka
    Antihistamine Substances. Tricyclic Analogues of N-(4,4-Diphenyl-3-butene-1-yl)nipecotic Acid and Some Related Compounds
    1994, Vol. 59, Issue 3, pp. 667–674 [Abstract]
  • Alexandra Šilhánková, Karel Dobrovský, Ivan Krejčí and Zdeněk Polívka
    Compounds Interacting with the Neuroexcitatory Amino Acids: Synthesis of 2-(4-Aralkylpiperazine-1-yl)-1-arylethanols
    1994, Vol. 59, Issue 3, pp. 658–666 [Abstract]
  • Eva Klinotová, Jiří Klinot, Václav Křeček, Stanislav Hilgard, Miloš Buděšínský and Jan Malát
    Structure of Dimeric Compounds Obtained from 3β-Acetoxy-21,22-dioxo-18α,19βH-ursan-28,20β-olide
    1993, Vol. 58, Issue 7, pp. 1675–1691 [Abstract]
  • Urszula Rychłewska, Beata Szczepanska, Miloš Buděšínský, David Šaman, Soňa Vašíčková, Bohdan Drożdż, Halina Grabarczyk and Miroslav Holub
    Crystal Structure of the Native Sesquiterpene Lactone Arctolide
    1993, Vol. 58, Issue 4, pp. 909–917 [Abstract]
  • Jaroslav Píš, Jiří Hykl, Miloš Buděšínský and Juraj Harmatha
    Cyclic Phenylboronates of Ecdysteroids as Products of Regiospecific Reaction with Phenylboronic Acid
    1993, Vol. 58, Issue 3, pp. 612–618 [Abstract]
  • Eva Klinotová, Jiří Klinot, Václav Křeček, Miloš Buděšínský and Bohumil Máca
    21,22-Disubstituted 18α,19βH-Ursane Derivatives with Oxabicyclooctane System in Ring E
    1993, Vol. 58, Issue 1, pp. 173–190 [Abstract]
  • Juraj Bernát, Ladislav Kniežo, Gabriela Birošová, Miloš Buděšínský, Jaroslav Podlaha, Jana Podlahová and Jiří Novotný
    Reactions of PO(NCS)3 with 4-Hydroxy-1,3-dioxanes. Crystal Structure of rel-(2S,4R,5S,6S)-2,6-Diethyl-5-methyl-4-(N'-benzylthioureido)-1,3-dioxane
    1992, Vol. 57, Issue 6, pp. 1299–1313 [Abstract]
  • Ełżbieta Błoszyk, Urszula Rychłewska, Beata Szczepanska, Miloš Buděšínský, Bohdan Drożdż and Miroslav Holub
    Sesquiterpene Lactones of Ambrosia artemisiifolia L. and Ambrosia trifida L. Species
    1992, Vol. 57, Issue 5, pp. 1092–1102 [Abstract]
  • Karel Stránský, Marta Semerdžieva, Miroslav Otmar, Želimír Procházka, Miloš Buděšínský, Karel Ubik, Jitka Kohoutová and Ludvík Streinz
    Antifungal Antibiotic from the Mushroom Agrocybe aegerita (BRIG.) SING.
    1992, Vol. 57, Issue 3, pp. 590–603 [Abstract]
  • Václav Křeček, Miloš Buděšínský and Alois Vystrčil
    Preparation of 20R and 20S Acetylamino-30-norlupane Derivatives
    1992, Vol. 57, Issue 3, pp. 556–564 [Abstract]
  • Otto Exner and Miloš Buděšínský
    Carbon-13 Substituent-Induced Chemical Shifts: Monosubstituted Benzene Derivatives
    1992, Vol. 57, Issue 3, pp. 497–507 [Abstract]
  • Karel Šindelář, Vojtěch Kmoníček, Marta Hrubantová and Zdeněk Polívka
    Substituted N,N-Dimethyl-3-(phenylthio)- and -4-(phenylthio)benzylamines
    1992, Vol. 57, Issue 1, pp. 194–203 [Abstract]
  • Irena Valterová, Miloš Buděšínský and Jan Vrkoč
    Defensive substances from the frontal gland secretion of Nasutitermes nigriceps termite soldiers
    1991, Vol. 56, Issue 12, pp. 2969–2977 [Abstract]
  • Jindřich Jindřich, Miloslav Černý, Tomáš Trnka and Miloš Buděšínský
    The synthesis of 4-O-oligoethylene glycol derivatives of 1,6-anhydro-β-D-glucopyranose and crown-ethers formed by their intramolecular cyclization
    1991, Vol. 56, Issue 12, pp. 2950–2963 [Abstract]
  • Jan Sejbal, Jiří Klinot, Miloš Buděšínský and Jiří Protiva
    Functionalization of 3β,28-lupanediol diacetate with chromium(VI) oxide
    1991, Vol. 56, Issue 12, pp. 2936–2949 [Abstract]
  • Eva Klinotová, Václav Křeček, Jiří Klinot, Miloš Buděšínský, Jaroslav Podlaha, Jana Podlahová and Jiří Ječný
    An unusual reaction of a bridged triterpenoid α-diketone with acetic anhydride
    1991, Vol. 56, Issue 12, pp. 2917–2935 [Abstract]
  • Miroslav Protiva
    Fifty years in chemical drug research
    1991, Vol. 56, Issue 11, pp. 2501–2772 [Abstract]
  • Karel Šindelář, Jiří Holoubek, Emil Svátek, Jan Metyš, Hana Blehová and Zdeněk Polívka
    Potential antihistaminics: Tricyclic carboxylic acids derived from 6,11-dihydrodibenzo[b,e]thiepine and 4,9-dihydrothieno[2,3-c]-2-benzothiepine
    1991, Vol. 56, Issue 11, pp. 2482–2493 [Abstract]
  • Vojtěch Kmoníček, Josef Pomykáček, Jiří Holoubek, Emil Svátek, Martin Valchář, Jiřina Metyšová and Zdeněk Polívka
    Potential antidepressants: 2-(fluoro-, chloro-, bromo- and cyanophenylthio)benzylamines as inhibitors of 5-hydroxytryptamine and noradrenaline re-uptake in brain
    1991, Vol. 56, Issue 11, pp. 2468–2481 [Abstract]
  • Otto Exner and Miloš Buděšínský*
    Correlation of substituent – inducted chemical shifts of aromatic protons: Substituted benzonitriles and methyl benzoates
    1991, Vol. 56, Issue 11, pp. 2234–2250 [Abstract]
  • Jan Sejbal, Jiří Klinot and Miloš Buděšínský
    Photolyses and pyrolyses of triterpenoid nitrites
    1991, Vol. 56, Issue 8, pp. 1732–1743 [Abstract]
  • Vladimír Valenta, Marie Vlková, Martin Valchář, Karel Dobrovský and Zdeněk Polívka
    Potential antidepressants: 3-Aryl-3-(arylthio)propylamines as selective inhibitors of 5-hydroxytryptamine re-uptake in the brain
    1991, Vol. 56, Issue 7, pp. 1525–1533 [Abstract]
  • Miloš Buděšínský, Alexander Kasal, Želimír Procházka, Huynh Kim Thoa, Soňa Vašíčková and Pavel Kočovský
    Revision of the structure of 3-methoxy-14α-hydroxy-D-homo-1,3,5-(10)-estratrien-17a-one. A simple 1H NMR method for the determination of configuration of hydroxy group in position 5 and/or 14 of the D-homo-steroid skeleton
    1991, Vol. 56, Issue 7, pp. 1512–1524 [Abstract]
  • Zdeněk Arnold, Miloš Buděšínský and Magdalena Pánková
    Reactivity of triformylmethane. I. Reactions of triformylmethane with selected types of amino compounds
    1991, Vol. 56, Issue 5, pp. 1019–1031 [Abstract]
  • Alois Vystrčil, Václav Křeček, Jiří Protiva and Miloš Buděšínský
    Anhydrobetulin and its derivatives
    1991, Vol. 56, Issue 4, pp. 886–904 [Abstract]
  • Karel Šindelář, Josef Pomykáček, Jiří Holubek, Emil Svátek, Martin Valchář, Karel Dobrovský, Jiřina Metyšová and Zdeněk Polívka
    Potential antidepressants and selective inhibitors of 5-hydroxytryptamine re-uptake in the brain: Synthesis of several potential metabolites of moxifetin and of two A-ring fluorinated analogues
    1991, Vol. 56, Issue 2, pp. 459–477 [Abstract]
  • Karel Šindelář, Josef Pomykáček, Martin Valchář, Karel Dobrovský, Jiřina Metyšová and Zdeněk Polívka
    Potential antidepressants and inhibitors of 5-hydroxytryptamine and noradrenaline re-uptake in the brain: N,N-Dimethyl-(arylthio)thenylamines and N,N-dimethyl-2-(thienylthio)benzylamines
    1991, Vol. 56, Issue 2, pp. 449–458 [Abstract]
  • Miloš Buděšínský, Dan Johnels, Ulf Edlund and Otto Exner
    Carbon-13 substituent-induced chemical shifts in benzene derivatives: Substituted anilines
    1991, Vol. 56, Issue 2, pp. 368–385 [Abstract]
  • Vladimír Valenta, Jiří Holubek, Emil Svátek, Martin Valchář, Ivan Krejčí and Miroslav Protiva
    Potential nootropic agents: Synthesis of some (2-oxo-1-pyrrolidinyl)acetamides and some related compounds
    1990, Vol. 55, Issue 11, pp. 2756–2764 [Abstract]
  • Václav Černý and Miloš Buděšínský
    A route to 24-epibrassinolide from ergosterol avoiding the use of osmium tetroxide
    1990, Vol. 55, Issue 11, pp. 2738–2755 [Abstract]
  • Ivan Černý, Vladimír Pouzar, Miloš Buděšínský, Pavel Drašar and Miroslav Havel
    Epimeric 17-hydroxy derivatives of 14β-androst-5-en-3β-yl acetate
    1990, Vol. 55, Issue 10, pp. 2510–2520 [Abstract]
  • Zdeněk Vejdělek and Miroslav Protiva
    Synthetic experiments aiming at 1,2,4,5-tetrahydro-3-benzothiepin derivatives
    1990, Vol. 55, Issue 9, pp. 2351–2356 [Abstract]
  • Zdeněk Vejdělek and Miroslav Protiva
    Synthesis of some derivatives of 1-phenyl-2,3,4,5-tetrahydro-1H-3-benzazepine and 11-phenyl-5,6-dihydro-11H-s-triazolo[3,4-b]-3-benzazepine
    1990, Vol. 55, Issue 9, pp. 2345–2350 [Abstract]
  • Vladimír Valenta, Jiří Holubek, Emil Svátek and Miroslav Protiva
    Potential cholinergic and anticholinergic compounds: Synthesis of 2,8-substituted 2,8-diazaspiro[4,5]decane-1,3-diones
    1990, Vol. 55, Issue 9, pp. 2304–2316 [Abstract]
  • Karel Šindelář, Jiří Jílek, Josef Pomykáček, Vladimír Valenta, Marta Hrubantová, Marie Vlková, Jiří Holubek, Emil Svátek, Miroslav Ryska, Jiřina Metyšová and Miroslav Protiva
    Tricyclic neuroleptics: Synthesis of metabolites of isofloxythepin and some related compounds
    1990, Vol. 55, Issue 9, pp. 2282–2303 [Abstract]
  • Jiří Jílek, Miroslav Rajšner, Vladimír Valenta, Miloš Borovička, Jiří Holubek, Miroslav Ryska, Emil Svátek, Jan Metyš and Miroslav Protiva
    Synthesis of piperidine derivatives as potential analgetic agents
    1990, Vol. 55, Issue 7, pp. 1828–1853 [Abstract]
  • Vojtěch Kmoníček, Emil Svátek, Jiří Holubek, Miroslav Ryska, Martin Valchář and Miroslav Protiva
    Synthesis of 1-acyl- and 1-(thioacyl)-4-benzylpiperazines as potential antidepressants
    1990, Vol. 55, Issue 7, pp. 1817–1827 [Abstract]
  • Vladimír Valenta, Karel Šindelář, Jiří Holubek, Miroslav Ryska, Ivan Krejčí, Antonín Dlabač and Miroslav Protiva
    Potential nootropic agents: Synthesis of a series of (2-oxo-1-pyrrolidinyl)acetic acid piperazides
    1990, Vol. 55, Issue 6, pp. 1613–1629 [Abstract]
  • Vojtěch Kmoníček, Zdeněk Vejdělek and Miroslav Protiva
    Synthesis of a series of 5-methyl-1H-imidazole-4-ylmethyl sulfides
    1990, Vol. 55, Issue 6, pp. 1602–1612 [Abstract]
  • Karel Šindelář, Jiří Holubek, Ivan Koruna, Marta Hrubantová and Miroslav Protiva
    Modified syntheses of 2-(methylthio)-10-(2-(1-methyl-2-piperidinyl)ethyl)phenothiazine (thioridazine) and 1-(3-(2-(methylsulfonyl)-10-phenothiazinyl)propyl)-piperidine-4-carboxamide (metopimazine)
    1990, Vol. 55, Issue 6, pp. 1586–1601 [Abstract]
  • Irena Valterová, Miloš Buděšínský, Jan Vrkoč and Glenn D. Prestwich
    (8Z)-1(15),8(9)-Trinervitadien-3α-ol from Nasutitermes nigriceps termites. The revised structure for a deffense compound of Trinervitermes gratiosus termites
    1990, Vol. 55, Issue 6, pp. 1580–1585 [Abstract]
  • Sergazy M. Adekenov, Miloš Buděšínský, Metram A. Abdikalikov, Coblandy M. Turdybekov, David Šaman, Ełżbieta Błoszyk, Bohdan Drożdż and Miroslav Holub
    Sesquiterpenic lactones of the Inula caspica BLUME species
    1990, Vol. 55, Issue 6, pp. 1568–1579 [Abstract]
  • Ełżbieta Błoszyk, Miloš Buděšínský, Włodzimierz M. Daniewski, Eva Pešková, Bohdan Drożdż and Miroslav Holub
    Sesquiterpenic lactones of Inula aschersoniana JANKA var. aschersoniana species
    1990, Vol. 55, Issue 6, pp. 1562–1567 [Abstract]
  • Jan Ježek, Evgenii A. Makarov, Tamara A. Balashova, Miloš Buděšínský, Tatyana M. Andronova and Vadim T. Ivanov
    Synthesis of tetrasaccharide containing glycopeptides related to bacterial cell wall starting from free tetrasaccharide by the pentafluorophenyl ester method
    1990, Vol. 55, Issue 5, pp. 1326–1335 [Abstract]
  • Vladimír Valenta, Jiří Holubek, Emil Svátek, Oluše Matoušová, Jiřina Metyšová and Miroslav Protiva
    Potential neuroleptics of the orthopramide series; synthesis of heterocyclic 5-amino-2-methoxybenzamides and of some related compounds
    1990, Vol. 55, Issue 5, pp. 1297–1310 [Abstract]
  • Zdeněk Vejdělek and Miroslav Protiva
    Potential antidepressants and tranquillizers: Synthesis of some 9-(aminoalkoxy)-2,3,6,7-tetrahydro-1H,5H-benzo[ij] quinolizines and 1-(substituted amino)-3-(1-naphthoxy)-2-propanols
    1990, Vol. 55, Issue 5, pp. 1290–1296 [Abstract]
  • Miroslav Protiva, Vladimír Valenta, Zdeňka Kopicová, Juraj Lukáč, Jiří Holubek and Ivan Krejčí
    Potential cerebral stimulants: Esters of 2-dimethylaminoethanol with some lipophilic carboxylic acids
    1990, Vol. 55, Issue 5, pp. 1278–1289 [Abstract]
  • Jiří Jílek, Karel Šindelář, Jaroslava Grimová, Eva Maturová, Jiří Holubek, Emil Svátek, Jiřina Metyšová, Jan Metyš, Marta Hrubantová and Miroslav Protiva
    Potential antidepressant and anti-inflammatory agents: 4-(2-Propylthio)acetophenone oximes and 4-(2-propylthio)phenylalkanoic acids
    1990, Vol. 55, Issue 5, pp. 1266–1277 [Abstract]
  • Jiří Urban, Zdeněk Šedivý, Jiří Holubek, Emil Svátek, Miroslav Ryska, Ivan Koruna, Antonín Dlabač, Martin Valchář, Jiřina Metyšová, Zdeněk Polívka, Karel Šindelář, Josef Pomykáček, Marta Hrubantová and Miroslav Protiva
    Potential antidepressants: 1-(2-(Methoxy- and hydroxyphenylthio)phenyl)-2-propylamines
    1990, Vol. 55, Issue 4, pp. 1077–1098 [Abstract]
  • Vladimír Valenta, Zdeněk Vejdělek, Karel Šindelář and Miroslav Protiva
    Potential anticonvulsants: Some derivatives and analogues of 2-propylpentanoic acid
    1990, Vol. 55, Issue 4, pp. 1067–1076 [Abstract]
  • Miloš Beran, Antonín Černý, Miroslav Kuchař, Hana Adamírová, Jiří Holubek, Jan Taimr, Jaroslav Vachek, Maria Frühaufová, Karel Řežábek, Martin Valchář and Ivan Krejčí
    9,10-Dihydroergopeptines modified in position 6
    1990, Vol. 55, Issue 3, pp. 819–832 [Abstract]
  • Vladimír Valenta, Marie Vlková, Jiří Holubek, Emil Svátek, Jiřina Metyšová and Miroslav Protiva
    Potential neuroleptics of the orthopramide series; Synthesis of N-(3-(tert.amino)propyl)-5-sulfamoyl-2-methoxybenzamides
    1990, Vol. 55, Issue 3, pp. 797–808 [Abstract]
  • Karel Šindelář, Jiří Holubek, Emil Svátek, Jiří Schlanger, Antonín Dlabač, Martin Valchář, Marta Hrubantová and Miroslav Protiva
    Open-ring models of hetero-cannabinoids: Synthesis of 2-(alkylthio)-5-(2-aminoethyl)hydroquinone derivatives
    1990, Vol. 55, Issue 3, pp. 782–796 [Abstract]
  • Jiří Klinot, Miloš Buděšínský and Jarmil Světlý
    Conformation of ring A in triterpenoid and 4,4-dimethylsteroid 3-ketones. Chemical shifts of methyl protons and lanthanide and benzene induced shifts
    1990, Vol. 55, Issue 3, pp. 766–781 [Abstract]
  • Miroslav Kuchař, Jaroslava Grimová, Václav Rejholec, Hana Tomková, Magda Jelínková and Jiří Holubek
    Use of QSAR in design of antiinflammatory fluorinated arylalkanoic acids
    1990, Vol. 55, Issue 1, pp. 296–306 [Abstract]
  • Karel Šindelář, Vladimír Valenta, Jiří Holubek, Oluše Matoušová and Miroslav Protiva
    Potential antidepressants. Synthesis of 6,11-dihydrodibenzo[b,e]thiepin-11-yl (dimethylaminomethyl)phenyl ethers, sulfides, amines and some related compounds
    1990, Vol. 55, Issue 1, pp. 282–295 [Abstract]
  • Jiří Jílek, Karel Šindelář, Josef Pomykáček, Vojtěch Kmoníček, Zdeněk Šedivý, Marta Hrubantová, Jiří Holubek, Emil Svátek, Miroslav Ryska, Ivan Koruna, Martin Valchář, Antonín Dlabač, Jiřina Metyšová, Nataša Dlohožková and Miroslav Protiva
    Potential antidepressants: 2-(Methoxy- and hydroxyphenylthio)benzylamines as selective inhibitors of 5-hydroxytryptamine re-uptake in the brain
    1989, Vol. 54, Issue 12, pp. 3294–3338 [Abstract]
  • Jaroslav Podlaha, Miloš Buděšínský, Jana Podlahová and Jindřich Hašek
    Crystal and solution structure of (E)-1,2-bis(ethylsulphonyl)cyclobutane-1,2-dicarbonitrile
    1989, Vol. 54, Issue 12, pp. 3253–3259 [Abstract]
  • Marcela Krečmerová, Miloslav Černý, Miloš Buděšínský and Antonín Holý
    Utilization of 1,6-anhydrohexoses for the preparation of some aliphatic adenosine analogs
    1989, Vol. 54, Issue 10, pp. 2753–2766 [Abstract]
  • Zdeněk Polívka, Miloš Buděšínský, Jiří Holubek, Bohdan Schneider, Zdeněk Šedivý, Emil Svátek, Oluše Matoušová, Jan Metyš, Martin Valchář, Radomír Souček and Miroslav Protiva
    4H-Benzo[4,5]cyclohepta[1,2-b]thiophenes and 9,10-dihydro derivatives - Sulfonium analogues of pizotifen and ketotifen; Chirality of ketotifen; Synthesis of the 2-bromo derivative of ketotifen
    1989, Vol. 54, Issue 9, pp. 2443–2469 [Abstract]
  • Jiří Jílek, Jiří Urban, Vojtěch Kmoníček, Josef Pomykáček, Jiří Holubek, Emil Svátek, Oluše Matoušová, Jan Metyš, Martin Valchář, Stanislav Wildt and Miroslav Protiva
    Potential anticonvulsants: 3-Chlorobenzophenone derivatives
    1989, Vol. 54, Issue 8, pp. 2248–2260 [Abstract]
  • Karel Šindelář, Marta Hrubantová, Emil Svátek, Oluše Matoušová, Jiřina Metyšová, Martin Valchář and Miroslav Protiva
    Potential antidepressants: 4-(Thioaryloxy)piperidines
    1989, Vol. 54, Issue 8, pp. 2240–2247 [Abstract]
  • Jiří Jílek, Jiří Urban, Petr Taufmann, Jiří Holubek, Antonín Dlabač, Martin Valchář and Miroslav Protiva
    Potential antidepressants: 2-(Phenylthio)aralkylamines
    1989, Vol. 54, Issue 7, pp. 1995–2008 [Abstract]
  • Vladimír Valenta, Marie Vlková, Jiří Holubek, Jiřina Metyšová and Miroslav Protiva
    Potential antidepressants: 10-Amino-2-chloro-10,11-dihydrodibenzo[b,f]thiepins
    1989, Vol. 54, Issue 7, pp. 1979–1994 [Abstract]
  • Irena Červená, Jiří Holubek, Emil Svátek, Jan Metyš and Miroslav Protiva
    Potential antidepressants: 2-(Aminoalkoxy)biphenyls and some related ω-substituted 2-alkoxybiphenyls
    1989, Vol. 54, Issue 7, pp. 1966–1978 [Abstract]
  • Irena Červená, Jiří Holubek, Emil Svátek, Miroslav Ryska and Miroslav Protiva
    Potential antidepressants: 6-(Aminoalkoxy)dibenzo[b,f]thiepin-10(11H)-ones and 6-(aminoalkoxy)-10,11-dihydrodibenzo[b,f]thiepin-10-ols
    1989, Vol. 54, Issue 7, pp. 1955–1965 [Abstract]
  • Miloš Buděšínský and Jiří Klinot
    Conformation of ring A in triterpenoid ketones. Carbon-13 chemical shifts and spin-lattice relaxation times of lupane and 18α-oleanane derivatives
    1989, Vol. 54, Issue 7, pp. 1928–1939 [Abstract]
  • Miloš Buděšínský, Halina Grabarczyk, Włodzimierz M. Daniewski, Andrzej Wawrzuń, Maria Gulumka, David Šaman, Bohdan Drożdż and Miroslav Holub
    Sesquiterpene lactones from Venidium hirsutum BEROL. species
    1989, Vol. 54, Issue 7, pp. 1919–1927 [Abstract]
  • Ełżbieta Błoszyk, Aleksandra Dudek, Zofia Kosturkiewicz, Urszula Rychłewska, Włodzimierz M. Daniewski, Maria Gulumka, Jan Nawrot, Miloš Buděšínský, Soňa Vašíčková and Miroslav Holub
    Sesquiterpene lactones of Cephalophora aromatica (HOOK.) SCHRADER and their deterrent activity. The stereostructure of geigerinin
    1989, Vol. 54, Issue 7, pp. 1903–1918 [Abstract]
  • Martin Mandel, Ludvík Novák, Miroslav Rajšner, Jiří Holubek and Vladislava Holá
    New synthesis of oxime-type beta-lactam antibiotics
    1989, Vol. 54, Issue 6, pp. 1734–1745 [Abstract]
  • Vojtěch Kmoníček, Zdeněk Vejdělek, Jiří Holubek, Martin Valchář and Miroslav Protiva
    Potential antidepressants: 1-(4-Aminoalkoxy)phenyl)-2-propylamines
    1989, Vol. 54, Issue 6, pp. 1721–1733 [Abstract]
  • Vladimír Valenta, Marie Vlková and Miroslav Protiva
    Potential neurotropic and antiinflammatory agents: 2-Chloro-10,11-dihydrodibenzo[b,f]thiepin-10-yl sulfides
    1989, Vol. 54, Issue 5, pp. 1403–1421 [Abstract]
  • Hana Hulinská, Miroslav Ryska, Ivan Koruna, Jiří Holubek, Jan Taimr, Emil Svátek and Miroslav Protiva
    Some further 2-(4-substituted 1-piperazinyl)acetamides derived from 6,11-dihydrodibenzo[b,e]thiepin. Transformations of 6,11-dihydrodibenzo[b,e]thiepin derivatives into anthraquinones, anthrones and anthracenes
    1989, Vol. 54, Issue 5, pp. 1388–1402 [Abstract]
  • Hana Hulinská, Miloš Buděšínský, Jiří Holubek, Oluše Matoušová, Hana Frycová and Miroslav Protiva
    Reactions of N-substituted 2-aminopyridines with chloroacetyl chloride; Formation of a new series of heterocyclic betaines: 1-Substituted 4-chloromethyl-2-oxopyrido[1,2-a]pyrimidin-5-ium-3-olates
    1989, Vol. 54, Issue 5, pp. 1376–1387 [Abstract]
  • Jan Sejbal, Eva Klinotová, Markéta Bludská, Jiří Klinot and Miloš Buděšínský
    Conversion of betulin into careyagenolide (2α,3β-dihydroxy-18α,19βH-ursan-28,20β-olide)
    1989, Vol. 54, Issue 4, pp. 1036–1042 [Abstract]
  • Jiří Protiva, Václav Křeček, Bohumil Máca, Jiří Urban, Miloš Buděšínský and Miloš Procházka
    Synthesis of 4-(N-acetyl-L-tyrosyl)amino-2-iodobenzoic acid
    1989, Vol. 54, Issue 4, pp. 1012–1018 [Abstract]
  • Miloš Buděšínský, Le Viet Ngoc Phuong, Nestor Perez Souto, Włodzimierz M. Daniewski, Andrzej Wawrzuń, Maria Gumułka, Soňa Vašíčková, David Šaman, Bohdan Drożdż, Halina Grabarczyk, Urszula Rychłewska and Miroslav Holub
    Isolation and structures of sesquiterpene lactones: Aerial parts of Arctotis grandis THUNB. species
    1989, Vol. 54, Issue 2, pp. 473–486 [Abstract]
  • Jiří Klinot, Jiří Liška, Alena Forgáčová, Miloš Buděšínský, Jiří Protiva, Stanislav Hilgard and Alois Vystrčil
    Acid-catalyzed rearrangements of an A(1)-nor-triterpenoid 2α,3α-epoxide
    1989, Vol. 54, Issue 2, pp. 413–429 [Abstract]
  • Zdeněk Polívka, Vladimír Valenta, Karel Šindelář, Jiří Holubek, Miloš Buděšínský, Miroslav Ryska, Ivan Koruna, Jitka Kohoutová, Jan Metyš, Jiřina Metyšová, Martin Valchář and Miroslav Protiva
    Potential antidepressants: Saturated side chain amines derived from 6,11-dihydrodibenzo[b,e]thiepin and 4,9-dihydrothieno[2,3-c]-2-benzothiepin
    1989, Vol. 54, Issue 1, pp. 235–247 [Abstract]
  • Karel Šindelář, Jiřina Metyšová and Miroslav Protiva
    Potential antidepressants: 2-(6,11-Dihydrodibenzo[b,e]thiepin-11-yl)-4,5-dihydroimidazoles
    1989, Vol. 54, Issue 1, pp. 229–234 [Abstract]
  • Irena Červená, Jiří Holubek, Emil Svátek, Jan Metyš, Martin Valchář and Miroslav Protiva
    Potential antidepressants: Synthesis of two 4-(aminoalkoxy)dibenzo[b,e]thiepin-11(6H)-ones
    1989, Vol. 54, Issue 1, pp. 225–228 [Abstract]
  • Miloš Buděšínský, David Šaman, Jan Pelnař, Soňa Vašíčková, Bohdan Drożdż, Halina Grabarczyk, Le Viet Ngoc Phuong and Miroslav Holub
    Arctolide-revision of its stereostructure and determination of absolute configuration. Detailed 1H and 13C NMR analysis
    1989, Vol. 54, Issue 1, pp. 166–188 [Abstract]
  • Jan Ježek, Milan Zaoral, Miloš Buděšínský, Jiří Günther and Jiří Rotta
    Muramyl-dipeptide analogues: Synthesis and biological activities
    1988, Vol. 53, Issue 11, pp. 2897–2906 [Abstract]
  • Jiří Jílek, Martin Valchář, Jiří Holubek, Nataša Dlohožková, Josef Pomykáček, Oluše Matoušová, Jiřina Metyšová and Miroslav Protiva
    Noncataleptic neuroleptic agents: 2-(4-(2-(2-Chloro-10,11-dihydrodibenzo[b,f]thiepin-10-yloxy)ethyl)piperazine-1-yl)ethanol and some related compounds
    1988, Vol. 53, Issue 11, pp. 2731–2741 [Abstract]
  • Zdena Koblicová, Jiří Holubek and Jan Trojánek
    Synthesis of stereoisomeric vincamines
    1988, Vol. 53, Issue 11, pp. 2722–2730 [Abstract]
  • Zdenko Procházka, Juris E. Ancans, Jiřina Slaninová, Alena Machová, Tomislav Barth, Jana Škopková, Miloš Buděšínský, Františka Pavlíková and Michal Lebl
    Synthesis and properties of analogues of vasopressin with 1-aminocyclopropane-1-carboxylic acid in position 9
    1988, Vol. 53, Issue 11, pp. 2604–2616 [Abstract]
  • Jan Hlaváček, Ivo Frič, Miloš Buděšínský and Karel Bláha
    An alternative route to Nα-methylamino acid derivatives: Synthesis and conformation of some Nα-acetyl-Nα-methylamino acid methylamides
    1988, Vol. 53, Issue 11, pp. 2473–2494 [Abstract]
  • Petr Maloň, C. L. Barness, Miloš Buděšínský, Rina K. Dukor, Dick Van der Helm, Timothy A. Keiderling, Zdena Koblicová, Františka Pavlíková, Miloš Tichý and Karel Bláha
    (1S,7S)-7-Methyl-6,9-diazatricyclo[6,3,0,01,6]tridecane-5,10-dione, a tricyclic spirodilactam containing non-planar amide groups: Synthesis, NMR, crystal structure, absolute configuration, electronic and vibrational circular dichroism
    1988, Vol. 53, Issue 11, pp. 2447–2472 [Abstract]
  • Miroslav Kuchař, Eva Maturová, Bohumila Brunová, Jaroslava Grimová, Hana Tomková and Jiří Holubek
    Quantitative relations between structure and antiinflammatory activity of aryloxoalkanoic acids
    1988, Vol. 53, Issue 8, pp. 1862–1872 [Abstract]
  • Hana Hulinská, Zdeněk Polívka, Jiří Jílek, Karel Šindelář, Jiří Holubek, Emil Svátek, Oluše Matoušová, Miloš Buděšínský, Hana Frycová and Miroslav Protiva
    Experimental antiulcer agents: N-substituted 2-(4-methyl-1-piperazinyl)acetamides as pirenzepine models and some related compounds
    1988, Vol. 53, Issue 8, pp. 1820–1844 [Abstract]
  • Zdeněk Polívka, Jan Metyš and Miroslav Protiva
    6,11-Dihydrodibenzo[b,e]thiepin-11-yl 3-quinuclidinyl ethers: New potential intidepressants and antihistamine agents
    1988, Vol. 53, Issue 8, pp. 1806–1811 [Abstract]
  • Václav Černý, Miloš Buděšínský, Miloš Ryba and František Tureček
    A contribution to peroxy acid oxidation of α,β-unsaturated ketones and linearly conjugated dienones: Reactions in the cholestane series
    1988, Vol. 53, Issue 7, pp. 1549–1567 [Abstract]
  • Irena Červená, Jiří Holubek, Emil Svátek and Miroslav Protiva
    Potential antidepressants: 4-(Aminoalkoxy)thioxanthones
    1988, Vol. 53, Issue 6, pp. 1307–1316 [Abstract]
  • Zdeněk Polívka, Jiřina Metyšová, Martin Valchář and Miroslav Protiva
    Potential antidepressants: N-phenacyl derivatives of (E)-N-methyl-3-(6,11-dihydrodibenzo[b,e]thiepin-11-ylidene)propylamine
    1988, Vol. 53, Issue 4, pp. 884–888 [Abstract]
  • Jiří Jílek, Jiří Holubek, Emil Svátek, Jan Metyš, Hana Frycová, Josef Pomykáček and Miroslav Protiva
    Tricyclic analogues of the antiallergic agent oxatomide: 1-(3-(4-(10,11-Dihydro-5H-dibenzo[a,d]cycloheptene-5-yl)-1-piperazinyl)propyl)-1,3-dihydro-2H-benzimidazol-2-one and the related 6,11-dihydrodibenzo[b,e]thiepin, 4,9-dihydrothieno[2,3-c]-2-benzothiepin, and 10,11-dihydrodibenzo[b,f]thiepin derivatives
    1988, Vol. 53, Issue 4, pp. 870–883 [Abstract]
  • Vladimír Valenta, Hana Hulinská, Jiří Holubek, Antonín Dlabač, Jan Metyš, Hana Frycová and Miroslav Protiva
    N-substituted derivatives of 6,11-dihydrodibenzo[b,e]thiepin-11-amine and related compounds; Synthesis and pharmacological screening
    1988, Vol. 53, Issue 4, pp. 860–869 [Abstract]
  • Karel Šindelář, Zdeněk Šedivý, Marta Hrubantová, Martin Valchář, Jiřina Metyšová and Miroslav Protiva
    Synthesis of (2-(phenylthio)phenyl)acetamidines and related amidoximes as potential antidepressants
    1988, Vol. 53, Issue 2, pp. 381–388 [Abstract]
  • Hana Hulinská, Petr Taufmann, Hana Frycová and Miroslav Protiva
    1-Methyl-, 1-phenyl-, and 1-(2-(2-dimethylaminoethoxy)-phenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole and their 2-substituted derivatives: Synthesis and pharmacological screening
    1988, Vol. 53, Issue 2, pp. 373–380 [Abstract]
  • Zdeněk Vejdělek, Jiří Holubek, Miloš Buděšínský, Miroslav Ryska, Emil Svátek and Miroslav Protiva
    Reactions of 4-chloro-1-nitrobenzene with (3-chloro-4-methoxyphenyl)acetonitrile and (3,4-dimethoxyphenyl)acetonitrile; Synthesis of 8-chloro-1-methyl (and methylthiomethyl-6-(3,4-disubstituted phenyl)-4H-s-triazolo[4,3-a]-1,4-benzodiazepines
    1988, Vol. 53, Issue 2, pp. 361–372 [Abstract]
  • Karel Šindelář, Jiří Holubek, Oluše Matoušová, Emil Svátek, Martin Valchář, Antonín Dlabač, Nataša Dlohožková, Marta Hrubantová and Miroslav Protiva
    Aminoalkylidene and aminoalkyl derivatives of 6,11-dihydrodibenzo[b,e]thiepin-2- and -9-carbonitrile and 4,10-dihydrothieno[2,3-c]-1-benzothiepin-6-carbonitrile; Antidepressants with a new activity profile
    1988, Vol. 53, Issue 2, pp. 340–360 [Abstract]
  • Zdeněk Vejdělek, Jan Metyš, Jiří Holubek, Miloš Buděšínský, Emil Svátek, Oluše Matoušová and Miroslav Protiva
    Potentional anxiolytics and hypnotics: 1-(Alkanesulfonamidoalkyl)-6-aryl-8-halogeno-s-triazolo[4,3-a]-1,4-benzodiazepines and related compounds
    1988, Vol. 53, Issue 1, pp. 132–144 [Abstract]
  • Vladimír Valenta, Jiří Holubek, Emil Svátek and Miroslav Protiva
    Synthesis of 4-methoxyphenoxyacetic and 3,4,5-trimethoxyphenoxyacetic acid amides and hydrazides as potential neurotropic and cardiovascular agents
    1987, Vol. 52, Issue 12, pp. 3013–3023 [Abstract]
  • Dalimil Dvořák, David Šaman, Miloš Buděšínský and Zdeněk Arnold
    Arbuzov rearrangement in the reaction of arylmethylenemalonaldehydes with trimethyl phosphite: Formation of 2-(α-dimethoxyphosphonylbenzyl)-3-methoxyacroleins
    1987, Vol. 52, Issue 12, pp. 2926–2935 [Abstract]
  • Irena Červená, Jiří Holubek, Emil Svátek, Martin Valchář and Miroslav Protiva
    Potential antidepressants: 3-Methyl-6-dimethylamino-1,2-diphenylhexan-3-ol and related compounds
    1987, Vol. 52, Issue 10, pp. 2564–2571 [Abstract]
  • Zdeněk Vejdělek, Jiří Holubek, Miroslav Ryska, Ivan Koruna, Emil Svátek, Miloš Buděšínský and Miroslav Protiva
    Reactions of 4-chloro-1-nitrobenzene with o-substituted phenylacetonitriles; Synthesis of 8-chloro-1-methyl(and methylthiomethyl)-6-(2-substituted phenyl)-4H-s-triazolo[4,3-a]-1,4-benzodiazepines
    1987, Vol. 52, Issue 10, pp. 2545–2563 [Abstract]
  • Vladimír Valenta, Jiří Holubek, Emil Svátek, Vladimír Miller, Marie Vlková and Miroslav Protiva
    2-Diethylaminoethyl esters of 1,3-disubstituted propane-2-carboxylic acids
    1987, Vol. 52, Issue 10, pp. 2534–2544 [Abstract]
  • Zdeněk Wimmer, Miloš Buděšínský, Tomáš Macek, Aleš Svatoš, David Šaman, Soňa Vašíčková and Miroslav Romaňuk
    Biotransformation of 2-(4-methoxybenzyl)-1-cyclohexanone by means of Saccharomyces cerevisiae
    1987, Vol. 52, Issue 9, pp. 2326–2337 [Abstract]
  • Karel Bláha, Miloš Buděšínský, Ivo Frič, Jan Pospíšek and Jindřich Symerský
    Conformation of diastereoisomeric cyclo(neopentylglycyl-prolyls): NMR, X-ray, and CD studies
    1987, Vol. 52, Issue 9, pp. 2295–2308 [Abstract]
  • Karel Šindelář, Miloš Buděšínský, Tomáš Vaněk, Jiří Holubek, Emil Svátek, Oluše Matoušová, Charles Wayne Rees and Miroslav Protiva
    Reaction of 6,11-dihydrodibenzo[b,e]thiepin-11-carbonitrile with 1,2-dibromoethane, a reinvestigation. Formation of 11,12-dihydro-6H-6,12-methanodibenzo[b,f]thiocin-12-carbonitrile
    1987, Vol. 52, Issue 9, pp. 2281–2294 [Abstract]
  • Vladimír Valenta and Miroslav Protiva
    Potential neuroleptics of the orthopramide series; Synthesis of N-substituted 5-(aminosulfonyl)-2-methoxybenzamides
    1987, Vol. 52, Issue 8, pp. 2095–2106 [Abstract]
  • Zdeněk Vejdělek and Miroslav Protiva
    1-(4-Cyclopentylphenyl)piperazine and its 4-substituted derivatives; Synthesis and biological screening
    1987, Vol. 52, Issue 7, pp. 1834–1840 [Abstract]
  • Miroslav Protiva, Jiří Jílek, Miroslav Rajšner, Karel Šindelář, Václav Bártl, Miroslav Ryska, Ivan Koruna, Jiří Holubek, Emil Svátek, Jiřina Metyšová, Antonín Dlabač, Josef Pomykáček and František Mikšík
    Fluorinated tricyclic neuroleptics with prolonged action: derivatives and analogues of 2-(4-(7-fluoro-2-isopropyl-10,11-dihydrodibenzo[b,f]thiepin-11-yl)-piperazine-1-yl)ethanol
    1987, Vol. 52, Issue 7, pp. 1811–1833 [Abstract]
  • Ladislav Novotný, Miloš Buděšínský, Josef Jizba, Juraj Harmatha, Vít Lukeš, Wolfgang Lindner, Rolf Grosser and Günther Snatzke
    Configuration of natural 9-hydroxyfuroeremophilane, its 9-hydroxy epimer and furanopetasin: NMR and CD studies
    1987, Vol. 52, Issue 7, pp. 1786–1802 [Abstract]
  • Zdeněk Polívka, Irena Lichá, Petr Taufmann, Emil Svátek, Jiří Holubek and Miroslav Protiva
    Synthesis of 3-(6,11-dihydrodibenzo[b,e]thiepin-11-ylidene)propanoic acid and related compounds
    1987, Vol. 52, Issue 6, pp. 1566–1582 [Abstract]
  • Jiří Urban, Emil Svátek, Miroslav Ryska, Jan Metyš, Stanislav Wildt and Miroslav Protiva
    4-Aryl-3-(dimethylaminomethyl)thiacyclohexan-4-ols including the thia analogue of tramadol; Synthesis and analgetic activity
    1987, Vol. 52, Issue 5, pp. 1340–1351 [Abstract]
  • Zdeněk Vejdělek and Miroslav Protiva
    4-Amino-1-(4-cyclopentylphenyl)butan-1-ones; Synthesis and biological screening
    1987, Vol. 52, Issue 4, pp. 1073–1078 [Abstract]
  • Vladimír Valenta, Jiří Holubek and Miroslav Protiva
    4-Substituted 1-(1-(2-(arylthio)-5-halogenophenyl)ethyl)piperazines; Synthesis and biological screening
    1987, Vol. 52, Issue 4, pp. 1062–1072 [Abstract]
  • Vojtěch Kmoníček, Jiří Holubek, Emil Svátek, Jiřina Metyšová and Miroslav Protiva
    2-(tert.amino)-11-(4-methylpiperazino)dibenzo[b,f]thiepins and their 10,11-dihydro derivatives; Synthesis and neuroleptic activity
    1987, Vol. 52, Issue 3, pp. 793–803 [Abstract]
  • Silvio Cerrini, Doriano Lamba, Irena Valterová, Miloš Buděšínský, Jan Vrkoč and František Tureček
    Methyl 3α,6α-diacetoxy-10-oxo-(7α)-kemp-11-en-20-oate: The revised structure for the kempane derivative from the frontal gland secretion of Nasutitermes costalis soldiers
    1987, Vol. 52, Issue 3, pp. 707–713 [Abstract]
  • Miloš Buděšínský and David Šaman
    Identification of acyl groups occurring in sesquiterpene lactones: Proton and carbon-13 NMR study
    1987, Vol. 52, Issue 2, pp. 453–475 [Abstract]
  • Zdeněk Veselý, Jiří Holubek and Jan Trojánek
    Reactions in the series of substituted isoindolo[1,2-b][3]-benzazepin-5-ones
    1987, Vol. 52, Issue 1, pp. 233–241 [Abstract]
  • Miroslav Kuchař, Bohumila Brunová, Jaroslava Grimová, Stanislav Vaněček and Jiří Holubek
    Synthesis of cyclohexylaliphatic acids and their pharmacological properties
    1986, Vol. 51, Issue 12, pp. 2896–2908 [Abstract]
  • Irena Valterová, Soňa Vašíčková, Miloš Buděšínský and Jan Vrkoč
    Constituents of frontal gland secretion of peruvian termites Nasutitermes ephratae
    1986, Vol. 51, Issue 12, pp. 2884–2895 [Abstract]
  • Jiří Klinot, Jarmil Světlý, Eva Klinotová, Miloš Buděšínský and Alois Vystrčil
    Preparation of isomeric 2-methyl-1-oxotriterpenoids of the 18α-oleanane series; Conformation of ring A
    1986, Vol. 51, Issue 12, pp. 2869–2878 [Abstract]
  • Karel Šindelář, Jiří Holubek, Miroslav Ryska, Ivan Koruna and Miroslav Protiva
    5-Substituted and 5,7-disubstituted 5,7-dihydrodibenzo[c,e]thiepins and the corresponding S-oxygenated compounds: Alkylamines, carboxylic acids, and carboxamides; synthesis and pharmacological screening
    1986, Vol. 51, Issue 12, pp. 2848–2868 [Abstract]
  • Miroslav Protiva, Jiří Jílek, Irena Červená, Josef Pomykáček, Václav Bártl, Antonín Dlabač, Martin Valchář, Jiřina Metyšová, Jiří Holubek and Emil Svátek
    Noncataleptic neuroleptic agents: 4-Substituted 1-(2-chloro-7-fluoro-10,11-dihydrodibenzo[b,f]thiepin-10-yl)piperazines and related compounds
    1986, Vol. 51, Issue 11, pp. 2598–2616 [Abstract]
  • Ludvík Streinz, Irena Valterová, Zdeněk Wimmer, Miloš Buděšínský, David Šaman, Jitka Kohoutová, Miroslav Romaňuk and Jan Vrkoč
    Direct esterification of α-methoxy-α-(trifluoromethyl)phenylacetic acid
    1986, Vol. 51, Issue 10, pp. 2207–2213 [Abstract]
  • Zdeněk Polívka, Jan Metyš and Miroslav Protiva
    Heterocyclic ethers derived from 6,11-dihydrodibenzo[b,e]thiepin-11-ols and 4,9-dihydrothieno[2,3-c]-2-benzothiepin-4-ol; A new series of potential antidepressants and antihistamine agents
    1986, Vol. 51, Issue 9, pp. 2034–2049 [Abstract]
  • Włodzimierz M. Daniewski, Wojciech Kroszczyṅski, Ełżbieta Błoszyk, Bohdan Drożdż, Jan Nawrot, Urszula Rychłewska, Miloš Buděšínský and Miroslav Holub
    Sesquiterpenoids from Dittrichia viscosa (L.) GREUTER. Their structure and deterrent activity
    1986, Vol. 51, Issue 8, pp. 1710–1721 [Abstract]
  • Urszula Rychłewska, Derek J. Hodgson, Halina Grabarczyk, Bohdan Drożdż, Włodzimierz M. Daniewski, Wojciech Kroszczyṅski, Miloš Buděšínský and Miroslav Holub
    Sesquiterpene lactones of Urospermum dalechampii SCHMIDT
    1986, Vol. 51, Issue 8, pp. 1698–1709 [Abstract]
  • Jiří Jílek, Martin Valchář, Josef Pomykáček, Antonín Dlabač and Miroslav Protiva
    Noncataleptic neuroleptic agents: Synthesis of some esters of 2-chloro-10-(4-(2-hydroxyethyl)piperazino)-10,11-dihydrodibenzo[b,f]thiepin
    1986, Vol. 51, Issue 7, pp. 1503–1508 [Abstract]
  • Zdeněk Vejdělek and Miroslav Protiva
    N-(piperazinoacyl) and N-(piperazinoalkyl) derivatives of 4-cyclopentylaniline and related compounds: Synthesis and pharmacological screening
    1986, Vol. 51, Issue 7, pp. 1494–1502 [Abstract]
  • Zdeněk Vejdělek, Jiří Němec and Miroslav Protiva
    Synthesis of N-(1-phenyl-2-propyl)-2,5-diphenylpentylamine and some related compounds as potential neurotropic and cardiovascular drugs
    1986, Vol. 51, Issue 7, pp. 1487–1493 [Abstract]
  • Zdenka Smítalová, Miloš Buděšínský, David Šaman and Miroslav Holub
    Minor sesquiterpenic lactones of Laser trilobum (L) BORKH. species
    1986, Vol. 51, Issue 6, pp. 1323–1339 [Abstract]
  • Miloš Buděšínský, Antonín Trka, Karel Stránský and Milan Streibl
    Heterocyclic nitrogen-containing compounds from the extract of the springtail Tetrodontophora bielanensis (WAGA)
    1986, Vol. 51, Issue 4, pp. 956–963 [Abstract]
  • Karel Stránský, Antonín Trka, Miloš Buděšínský and Milan Streibl
    Lipidic compounds from the extract of the springtail Tetrodontophora bielanensis (WAGA)
    1986, Vol. 51, Issue 4, pp. 948–955 [Abstract]
  • Vojtěch Kmoníček, Emil Svátek, Jiří Holubek and Miroslav Protiva
    Synthesis of potential neuroleptics and tranquillizers: 2-(tert.Amino)-9-(3-dimethylaminopropylidene)thioxanthenes
    1986, Vol. 51, Issue 4, pp. 937–947 [Abstract]
  • Miroslav Holub, Miloš Buděšínský, Zdenka Smítalová, David Šaman and Urszula Rychłewska
    Structure of isosilerolide, relative and absolute configuration of silerolide and lasolide - Sesquiterpenic lactones of new stereoisomeric type of eudesmanolides
    1986, Vol. 51, Issue 4, pp. 903–929 [Abstract]
  • Miroslav Protiva, Jiří Jílek, Miroslav Rajšner, Josef Pomykáček, Miroslav Ryska, Jiří Holubek, Emil Svátek and Jiřina Metyšová
    Fluorinated tricyclic neuroleptics with prolonged action: 7-Fluoro-11-[4-(2-hydroxyethyl)piperazino]-2-isopropyl-10,11-dihydrodibenzo[b,f]thiepin
    1986, Vol. 51, Issue 3, pp. 698–722 [Abstract]
  • Václav Křeček, Jiří Protiva, Miloš Buděšínský, Eva Klinotová and Alois Vystrčil
    Preparation of C(18)-empiric 20,29,30-trinorlupane derivatives. 1H, 13C NMR and mass spectra
    1986, Vol. 51, Issue 3, pp. 621–635 [Abstract]
  • Jiří Klinot, Miloš Buděšínský, Eva Klinotová and Alois Vystrčil
    Conformation of the A ring in 1-oxo and 3-oxotriterpenoids. Vicinal interproton coupling constants
    1986, Vol. 51, Issue 3, pp. 593–610 [Abstract]
  • Alois Vystrčil, Václav Křeček, Miloš Buděšínský and Jiří Protiva
    Isomeric oximes of 30-norlupan-20-one and its derivatives
    1986, Vol. 51, Issue 3, pp. 581–592 [Abstract]
  • Miroslav Protiva, Antonín Dlabač, Martin Valchář, Stanislav Wildt, Irena Červená and Zdeněk Šedivý
    Potential noncataleptic neuroleptic agents; 2,6-Dichloro-, 2,7-dichloro- and 2,8-dichloro-10-piperazino-10,11-dihydrodibenzo[b,f]thiepins
    1986, Vol. 51, Issue 1, pp. 156–166 [Abstract]
  • Irena Červená, Jiří Holubek, Emil Svátek, Jiřina Metyšová, Martin Valchář, Antonín Dlabač, Stanislav Wildt and Miroslav Protiva
    6-Substituted and 2-chloro-6-substituted 10-piperazino-10,11-dihydrodibenzo[b,f]thiepins as potential antidepressants; Synthesis and pharmacology
    1986, Vol. 51, Issue 1, pp. 141–155 [Abstract]
  • Urszula Rychłewska, Derek J. Hodgson, Miroslav Holub, Miloš Buděšínský and Zdenka Smítalová
    The structure of 2-oxo-8α-angeloyloxy-11α-acetoxy-5βH,6αH,7αH-guai-1(10),3-dien-6,12-olide, a sesquiterpenic lactone from Laserpitium prutenicum L. revision of the stereostructures of native 2-oxoguai-1(10),3-dien-6,12-olides from the species of the Umbelliferae family
    1985, Vol. 50, Issue 11, pp. 2607–2624 [Abstract]
  • Dalimil Dvořák, Miloš Buděšínský, David Šaman and Zdeněk Arnold
    Benzylidenemalonaldehydes: A redox reaction during the attempted cycloaddition on nitrosobenzene
    1985, Vol. 50, Issue 10, pp. 2260–2264 [Abstract]
  • Jiří Jílek, Jiří Holubek, Emil Svátek, Jiřina Metyšová, Josef Pomykáček, Zdeněk Šedivý and Miroslav Protiva
    Potential metabolites of the neuroleptic agents belonging to the 8-methylthio-10-piperazino-10,11-dihydrodibenzo[b,f]thiepin series; Synthesis of 2-hydroxy and 3-hydroxy derivatives
    1985, Vol. 50, Issue 10, pp. 2179–2190 [Abstract]
  • Milena Masojídková, Jaroslav Zajíček, Miloš Buděšínský, Ivan Rosenberg and Antonín Holý
    Conformational study on ribonucleoside O-phosphonylmethyl derivatives by 1H NMR spectroscopy
    1985, Vol. 50, Issue 8, pp. 1899–1905 [Abstract]
  • Miroslav Protiva, Zdeněk Šedivý, Jiří Holubek, Emil Svátek and Jiří Němec
    Cyclic amidines derived from benz[c,d]indole and 4,5-dihydro-3H-1-benzazepine including some related compounds: Synthesis and pharmacological screening
    1985, Vol. 50, Issue 8, pp. 1888–1898 [Abstract]
  • Miroslav Holub, Miloš Buděšínský, Zdenka Smítalová, David Šaman and Urszula Rychłewska
    Structure of laserolide and isolaserolide: Revision of constitution and determination of relative and absolute configuration
    1985, Vol. 50, Issue 8, pp. 1878–1887 [Abstract]
  • Zdeněk Vejdělek, Václav Bártl, Emil Svátek and Miroslav Protiva
    Synthesis of several compounds related to 1-(4-methylsulfonylphenacyl)-4-phenylpiperazine and their pharmacological screening
    1985, Vol. 50, Issue 7, pp. 1498–1506 [Abstract]
  • Karel Šindelář, Jiří Holubek, Emil Svátek, Miroslav Ryska, Martin Valchář and Miroslav Protiva
    Butaclamol-like neuroleptic agents: Synthesis of 1-(11H-dibenz[b,f]-1,4-oxathiepin-11-yl)methyl-4-isobutylpiperidin-4-ol and of some related compounds
    1985, Vol. 50, Issue 7, pp. 1484–1497 [Abstract]
  • Karel Šindelář, Jan Metyš and Miroslav Protiva
    Potential antidiarrheal agents: 1-(11-Cyano-6,11-dihydrodibenzo[b,e]thiepin-11-yl-alkyl)- and 1-(10-cyano-10,11-dihydrodibenzo[b,f]thiepin-10-yl-alkyl)-4-substituted piperidines
    1985, Vol. 50, Issue 5, pp. 1089–1096 [Abstract]
  • Zdeněk Polívka, Jiří Holubek, Emil Svátek, Jan Metyš and Miroslav Protiva
    Synthesis of the semi-rigid analogues of prothiadene and dithiadene as potential antidepressant and antihistamine agents: 11-[2-(Dimethylaminomethyl)cyclohexylidene]-6,11-dihydrodibenzo[b,e]thiepins and 4-[2-(dimethylaminomethyl)cyclohexylidene]-4,9-dihydrothieno-[2,3-c]-2-benzothiepins
    1985, Vol. 50, Issue 5, pp. 1078–1088 [Abstract]
  • Vladimír Valenta, Zdeněk Prošek, Jiřina Metyšová, Martin Valchář, Antonín Dlabač and Miroslav Protiva
    Cataleptic and noncataleptic neuroleptic agents: Synthesis and pharmacology of 4-(2-chloro and 8-chloro substituted 10,11-dihydrodibenzo[b,f]thiepin-10-yl)piperazine-1-ylalkyl ethers and sulfides
    1985, Vol. 50, Issue 5, pp. 1070–1077 [Abstract]
  • Zdeněk Vejdělek, Zdeněk Polívka and Miroslav Protiva
    Synthesis of 7-chloro-5-(4-chlorophenyl)-1-methyl-1,3-dihydro-1,4-benzodiazepin-2-one
    1985, Vol. 50, Issue 5, pp. 1064–1069 [Abstract]
  • Jan Šmidrkal, Jiří Holubek and Jan Trojánek
    The synthesis of 2,3,7,8-bismethylenedioxy-11-methoxy-5-methylbenzo[c]phenanthridinium chloride
    1985, Vol. 50, Issue 4, pp. 984–990 [Abstract]
  • Jan Šmidrkal, Jiří Holubek, Jiří Šlanger and Jan Trojánek
    Attempts at the synthesis of 11-methoxysubstituted benzo[c]phenantridines
    1985, Vol. 50, Issue 4, pp. 861–868 [Abstract]
  • Jiří Jílek, Jiří Holubek, Emil Svátek, Jiří Schlanger, Josef Pomykáček and Miroslav Protiva
    Highly polar potential metabolites of the neuroleptic agent oxyprothepin: Synthesis of 2-hydroxy-8-methylsulfonyl and 3-hydroxy-8-methylsulfonyl derivatives of 10-[4-(3-hydroxypropyl)piperazino]-10,11-dihydrodibenzo[b,f]thiepin
    1985, Vol. 50, Issue 2, pp. 519–537 [Abstract]
  • Vladimír Valenta and Miroslav Protiva
    Synthesis of several 4-hydroxy-3,5-dimethoxybenzamides, their O-substituted derivatives and some related compounds as potential neurotropic agents
    1985, Vol. 50, Issue 2, pp. 510–518 [Abstract]
  • Karel Šindelář, Jiří Holubek, Jiří Schlanger, Antonín Dlabač, Martin Valchář and Miroslav Protiva
    Synthesis of spiro(piperidine-4,6'-dibenz[b,e]-1,4-oxathiepin) and its 1-methyl derivative as potential antidepressant agents
    1985, Vol. 50, Issue 2, pp. 503–509 [Abstract]
  • Wojciech Kroszczyṅski, Włodzimierz M. Daniewski, Miloš Buděšínský, David Šaman, Halina Grabarczyk, Bohdan Drożdż and Miroslav Holub
    Minor sesquiterpenic lactones from Ursinia anthemoides (L.) POIRET
    1985, Vol. 50, Issue 1, pp. 94–102 [Abstract]
  • Karel Konečný, Milan Streibl, Soňa Vašíčková, Miloš Buděšínský, David Šaman, Karel Ubik and Vlastimil Herout
    Constituents of the liverwort Bazzania trilobata of Czech origin
    1985, Vol. 50, Issue 1, pp. 80–93 [Abstract]
  • Antonín Černý, Jiří Křepelka, Viktor Zikán, Drahuše Vlčková, Jaroslav Vachek, Jiří Holubek, Karel Řežábek, Maria Frühaufová, Miroslav Šeda, Jana Chlebounová and Otakar Marhan
    Some 6-substituted 1-[(5R,8S,10R)-8-ergolinyl]-3,3-diethylureas
    1984, Vol. 49, Issue 12, pp. 2828–2836 [Abstract]
  • Urszula Rychłewska, Miroslav Holub, Miloš Buděšínský and Zdenka Smítalová
    Stereostructure of slovanolides: X-ray crystallography of the 3-oxo-4αH,8α-benzoyloxy-10β,11α-diacetoxyslovanolide
    1984, Vol. 49, Issue 12, pp. 2790–2800 [Abstract]
  • Zdeněk Vejdělek, Jan Metyš, Jiří Holubek, Emil Svátek and Miroslav Protiva
    Potential antiparkinsonic agents: Synthesis and pharmacology of some 4-fluoro-4'-halogen'benzhydryl 2-(N,N-disubstituted amino)ethyl ethers
    1984, Vol. 49, Issue 11, pp. 2649–2660 [Abstract]
  • Jiří Jílek, Miroslav Rajšner, Jiřina Metyšová, Josef Pomykáček and Miroslav Protiva
    Fluorinated tricyclic neuroleptics with prolonged action: 8-Alkyl derivatives of 3-fluoro-10-piperazino-10,11-dihydrodibenzo[b,f]thiepins
    1984, Vol. 49, Issue 11, pp. 2638–2648 [Abstract]
  • Karel Šindelář, Jiří Holubek, Miroslav Ryska, Antonín Dlabač, Martin Valchář, Jiřina Metyšová and Miroslav Protiva
    Tricyclic compounds containing two chalcogen atoms in the central seven-membered rings as potential drugs: Synthesis of 3-chloro-6-(1-methyl-4-piperidyl)-6H-dibenz[b,e]-1,4-oxathiepin and 6-oxodibenz[b,e]-1,4-oxathiepin-2-acetic acid
    1984, Vol. 49, Issue 11, pp. 2531–2540 [Abstract]
  • Václav Bártl, Karel Šindelář, Vladimír Valenta, Jiří Holubek, Emil Svátek, Jiří Schlanger, Antonín Dlabač, Jiřina Metyšová and Miroslav Protiva
    Potential antipsychotic agents: 2-Chloro- and 2-methyl-11-(2-piperazinoethoxy)-6,11-dihydrodibenzo[b,e]thiepins and some related compounds; Synthesis and pharmacology
    1984, Vol. 49, Issue 11, pp. 2520–2530 [Abstract]
  • Václav Bártl, Vojtěch Kmoníček, Zdeněk Šedivý, Emil Svátek, Jiří Protiva and Miroslav Protiva
    Thioxanthene derivatives of pharmacological interest: 1,2,4-Trichloro and 2,4,5,6-tetrachloro derivatives of 9-(3-dimethylaminopropylidene)thioxanthene
    1984, Vol. 49, Issue 10, pp. 2295–2308 [Abstract]
  • Irena Valterová, Miloš Buděšínský, František Tureček and Jan Vrkoč
    Minor diterpene components of the defense secretion from the frontal gland of soldiers of the species Nasutitermes costalis (HOLMGREN)
    1984, Vol. 49, Issue 9, pp. 2024–2039 [Abstract]
  • Václav Bártl, Emil Svátek, Antonín Dlabač, Stanislav Wildt and Miroslav Protiva
    11-(3-[4-(2-Hydroxyethyl)piperazino]propylidene)-6,11-dihydrodibenzo[b,e]thiepin, its 2-chloro derivative and some related compounds as potential antipsychotic agents; Synthesis and pharmacology
    1984, Vol. 49, Issue 8, pp. 1816–1826 [Abstract]
  • Václav Bártl, Jiří Jílek, Jiřina Metyšová, Martin Valchář, Antonín Dlabač, Stanislav Wildt and Miroslav Protiva
    Neuroleptic 2-chloro-11-(2-piperazineethoxy)-10,11-dihydrodibenzo[b,f]thiepins: Synthesis and pharmacology
    1984, Vol. 49, Issue 8, pp. 1810–1815 [Abstract]
  • Václav Bártl, Antonín Dlabač, Martin Valchář and Miroslav Protiva
    11-(4-Piperidylidene)-6,11-dihydrodibenzo[b,e]thiepins as potential antipsychotic agents; Synthesis and pharmacology
    1984, Vol. 49, Issue 8, pp. 1800–1809 [Abstract]
  • Vojtěch Kmoníček, Václav Bártl and Miroslav Protiva
    Thioxanthene derivatives with neurotropic activity; synthesis of 9-(3-dimethylaminopropylidene)-2-(methylthiomethyl)thioxanthene and of some related compounds
    1984, Vol. 49, Issue 7, pp. 1722–1730 [Abstract]
  • Miloš Buděšínský, Miroslav Holub, David Šaman, Zdenka Smítalová, Ayhan Ulubelen and Sevil Öksüz
    Structure of istanbulin A and istanbulin B - two sesquiterpenic lactones from Smyrnium olusatrum L.
    1984, Vol. 49, Issue 5, pp. 1311–1317 [Abstract]
  • Karel Šindelář, Jiří Holubek, Miroslav Ryska, Emil Svátek, Antonín Dlabač, Martin Valchář and Miroslav Protiva
    Analogues of the neuroleptic agent isobutaclamol: Stereoisomeric 3b,4,5,6,7,9,9a,10-octahydro-[1]benzothiepino[2,3,4-ed]pyrido[2,1-a]isoquinolin-5-ols and some related compounds
    1984, Vol. 49, Issue 4, pp. 1021–1038 [Abstract]
  • Irena Červená and Miroslav Protiva
    1-[2-(2-Hydroxymethylphenylthio)benzyl]-4-methylpiperzine and related compounds as potential antidepressants: Synthesis and pharmacological acreening
    1984, Vol. 49, Issue 4, pp. 1009–1020 [Abstract]
  • Vladimír Valenta, Antonín Dlabač, Martin Valchář and Miroslav Protiva
    α-Benzyldopamine and some related compounds: Synthesis and pharmacological screening
    1984, Vol. 49, Issue 4, pp. 1002–1008 [Abstract]
  • Jiří Urban, Antonín Dlabač, Martin Valchář and Miroslav Protiva
    Potential noncataleptic neuroleptic agents: 2,3-Dichloro-10-[4-(2-hydroxyethyl)piperazino]-10,11-dihydrobenzo[b,f]thiepin
    1984, Vol. 49, Issue 4, pp. 992–1001 [Abstract]
  • Ivan Černý, Vladimír Pouzar, Pavel Drašar, Miloš Buděšínský and Miroslav Havel
    Glucosylation of 5-androsten-3β-ol derivatives containing butenolide, furan or unsaturated ester moieties in the side chain
    1984, Vol. 49, Issue 4, pp. 881–891 [Abstract]
  • Zdenka Smítalová, Miloš Buděšínský, David Šaman, Soňa Vašíčková and Miroslav Holub
    Components of the extract from the underground parts of Laserpitium siler L. of slovenian origin, mainly sesquiterpenic lactones
    1984, Vol. 49, Issue 4, pp. 852–870 [Abstract]
  • Karel Bláha, Ahmed M. Farag, Dick VAN DER Helm, M. Bilayet Hossain, Miloš Buděšínský, Petr Maloň, Jorga Smolíková and Miloš Tichý
    Stereoisomeric chiral 2,9-diazabicyclo[4.4.0.]decane-3,10-diones as models of dipeptide grouping: Synthesis, X-ray, IR, NMR and cd studies
    1984, Vol. 49, Issue 3, pp. 712–742 [Abstract]
  • Zdenko Procházka, Michal Lebl, Tomislav Barth, Jan Hlaváček, Antonín Trka, Miloš Buděšínský and Karel Jošt
    Synthesis and properties of oxytocin analogues modified in the tripeptide side chain
    1984, Vol. 49, Issue 3, pp. 642–652 [Abstract]
  • Miloš Buděšínský, David Šaman, Gerard Nowak, Bohdan Drożdż and Miroslav Holub
    9α-Hydroxyparthenolide from Zoegea baldschuanica C. WINKL. and its absolute configuration
    1984, Vol. 49, Issue 3, pp. 637–641 [Abstract]
  • Zdeněk Polívka, Jiří Holubek, Emil Svátek, Jan Metyš and Miroslav Protiva
    Potential hypnotics and anxiolytics: Synthesis of 2-bromo-4-(2-chlorophenyl)-9-[4-(2-methoxyethyl)piperazino]-6H-thieno[3,2,4-triazolo[4,3-a]-1,4-diazepine and of some related compounds
    1984, Vol. 49, Issue 3, pp. 621–636 [Abstract]
  • Jiří Jílek, Josef Pomykáček, Jiří Holubek, Emil Svátek, Miroslav Ryska, Jiří Protiva and Miroslav Protiva
    Reactions of 4,4'-disubstituted diphenyl sulfides with chloroacetyl chloride and aluminium chloride
    1984, Vol. 49, Issue 3, pp. 603–620 [Abstract]
  • Miloš Tichý, Ahmed Farag, Miloš Buděšínský, Ludmila P. Otroshchenko, Tatjana A. Shibanova and Karel Bláha
    Isomeric oxatricyclodecanones with non-planar lactone groups: Synthesis, absolute configuration, NMR and X-ray study
    1984, Vol. 49, Issue 2, pp. 513–532 [Abstract]
  • Miloš Buděšínský, Miloslav Černý, Jitka Doležalová, Miloš Kulhánek, Josef Pacák and Milan Tadra
    4-Deoxy-4-fluoro-D-fructose: Preparation and structure
    1984, Vol. 49, Issue 1, pp. 267–274 [Abstract]
  • Jaroslav Zajíček, Miloš Buděšínský and Jiří Farkaš
    Conformational study of blocked pentofuranoses and their 1,5-anhydro derivatives by 1H NMR spectroscopy
    1984, Vol. 49, Issue 1, pp. 235–243 [Abstract]
  • Miroslav Kuchař, Bohumila Brunová, Václav Rejholc, Magda Jelínková, Jiří Holubek and Oldřich Němeček
    Quantitative relations between structure and activation of fibrinolysis in selected series of arylaliphatic acids
    1984, Vol. 49, Issue 1, pp. 122–136 [Abstract]
  • Zdeněk Polívka, Jiří Jílek, Jiří Holubek, Emil Svátek, Antonín Dlabač, Martin Valchář and Miroslav Protiva
    Noncataleptic neuroleptic agents: 2-Halogeno-8-isopropyl-10-piperazino-10,11-dihydrodibenzo[b,f,]thiepins
    1984, Vol. 49, Issue 1, pp. 86–109 [Abstract]
  • Zdeněk Polívka, Jiří Holubek, Jan Metyš, Zdeněk Šedivý and Miroslav Protiva
    Potential hypnotics and anxiolytics: 8-Chloro-6-(2-chlorophenyl)-1-[4-(2-methoxyethyl)piperazino]-methyl-4H-s-triazolo[4,3-a]-1,4-benzodiazepine and related compounds
    1983, Vol. 48, Issue 12, pp. 3433–3443 [Abstract]
  • Zdeněk Vejdělek and Miroslav Protiva
    Potential antitussives: Synthesis and pharmacology of a series of 1-[2-amino-2-(4-fluorophenyl)ethyl]-4-(2-benzoylpropyl)piperazines
    1983, Vol. 48, Issue 10, pp. 2977–2988 [Abstract]
  • Zdeněk Polívka, Martin Valchář and Miroslav Protiva
    Potential noncataleptic neuroleptic agents: Synthesis and pharmacology of 7-chloro-4-[4-(2-hydroxyethyl)piperazino]-4,5-dihydrothieno[2,3-b]-1-benzothiepin
    1983, Vol. 48, Issue 10, pp. 2970–2976 [Abstract]
  • Petr Maloň, Petr Pančoška, Miloš Buděšínský, Jan Hlaváček, Jan Pospíšek and Karel Bláha
    Chiroptical properties and conformation of N-acetyl-L-amino acids N'-methylamides with aliphatic side chains
    1983, Vol. 48, Issue 10, pp. 2844–2861 [Abstract]
  • Miloslav Černý, Jitka Doležalová, Jindra Mácová, Josef Pacák, Tomáš Trnka and Miloš Buděšínský
    Preparation of 3-deoxy-3-fluoro-D-mannose and corresponding hexitol
    1983, Vol. 48, Issue 9, pp. 2693–2700 [Abstract]
  • Zdeněk Polívka, Miroslav Ryska, Jiří Holubek, Emil Svátek, Jan Metyš and Miroslav Protiva
    Potential hypnotics and anxiolytics in the 4H-s-triazolo[4,3-a]-1,4-benzodiazepine series: 8-Chloro-6-(2-chlorophenyl)-1-[4-(2-methoxyethyl)piperazino]-4H-s-triazolo[4,3-a]-1,4-benzodiazepine and some related compounds
    1983, Vol. 48, Issue 8, pp. 2395–2410 [Abstract]
  • Karel Šindelář, Jiří Holubek, Miroslav Ryska, Emil Svátek, Jiří Urban and Miroslav Protiva
    11-(Dimethylaminoalkyl)-6,11-dihydrodibenzo[b,e]thiepin-11-carbonitriles and some related compounds
    1983, Vol. 48, Issue 7, pp. 1898–1909 [Abstract]
  • Alois Vystrčil, Václav Křeček and Miloš Buděšínský
    Elimination reaction of angular hydroxymethyl groups of 20(29)-lupene derivatives
    1983, Vol. 48, Issue 5, pp. 1499–1507 [Abstract]
  • Antonín Černý, Viktor Zikán, Drahuše Vlčková, Jan Beneš, Jiří Holubek, Karel Řežábek, Marie Aušková and Jiří Křepelka
    (5R,8S,10R)-6-Alkyl-8-ergolinecarboxylic acids and some of their derivatives
    1983, Vol. 48, Issue 5, pp. 1483–1488 [Abstract]
  • Zdeněk Vejdělek and Miroslav Protiva
    Synthesis of two 1-substituted 8-bromo-6-(2-chlorophenyl)-4H-s-triazolo[4,3-a]-1,4-benzodiazepines
    1983, Vol. 48, Issue 5, pp. 1477–1482 [Abstract]
  • Zdeněk Polívka, Jiří Holubek, Emil Svátek, Antonín Dlabač, Dušan Půček, Zdeněk Šedivý and Miroslav Protiva
    3-(4-Methylpiperazino)dibenzo[b,f]-1,2,4-triazolo[4,3-d]-1,4-thiazepine and its 6-chloro and 12-chloro derivatives; Synthesis and pharmacology
    1983, Vol. 48, Issue 5, pp. 1465–1476 [Abstract]
  • Vladimír Valenta, Jiří Holubek, Emil Svátek, Antonín Dlabač, Marie Bartošová and Miroslav Protiva
    α-(4-Tolyl)dopamine, derivatives and analogues; Synthesis and pharmacological screening
    1983, Vol. 48, Issue 5, pp. 1447–1464 [Abstract]
  • Jiří Křepelka, Vladimír Pouzar, Jiří Schlanger, Jiří Holubek, Jiří Körbl, Fedir Jančik and Rudolf Kotva
    Oxidative transformations of some pyrimidine derivatives into oxazolidine derivatives
    1983, Vol. 48, Issue 4, pp. 1212–1223 [Abstract]
  • Karel Šindelář, Jiří Holubek, Miroslav Ryska, Emil Svátek, Jiří Urban, Jaroslava Grimová, Irena Červená, Marta Hrubantová and Miroslav Protiva
    Dibenzo[b,f]thiepin-10-carbonitrile, its 10,11-dihydro derivative, some transformation products and related compounds
    1983, Vol. 48, Issue 4, pp. 1187–1211 [Abstract]
  • Václav Bártl, Jiří Holubek, Emil Svátek, Marie Bartošová and Miroslav Protiva
    Potential anticonvulsants: Substituted N-benzylidene derivatives of 10-(4-aminopiperazino)-10,11-dihydrodibenzo[b,f]thiepins
    1983, Vol. 48, Issue 4, pp. 1173–1186 [Abstract]
  • Vladimír Valenta, Jiří Němec and Miroslav Protiva
    Basic amides of 2,4,5-trichlorophenoxyacetic, 2,4,6-trimethylphenoxyacetic and 4-bromo-3,5-dimethylphenoxyacetic acid and some related compounds; Synthesis and pharmacological screening
    1983, Vol. 48, Issue 4, pp. 1089–1096 [Abstract]
  • Miroslav Kuchař, Václav Rejholec, Zdeněk Roubal and Oluše Matoušová
    The effects of lipophilicity on the inhibition of denaturation of serum albumin and on the activation of fibrinolysis observed with a series of benzyloxyarylaliphatic acids
    1983, Vol. 48, Issue 4, pp. 1077–1088 [Abstract]
  • Jiří Jílek, Josef Pomykáček, Zdeněk Prošek, Jiří Holubek, Emil Svátek, Jiřina Metyšová, Antonín Dlabač and Miroslav Protiva
    8-Chloro and 8-methylthio derivatives of 10-piperazino-10,11-dihydrodibenzo[b,f]thiepins; New compounds and new procedures
    1983, Vol. 48, Issue 3, pp. 906–927 [Abstract]
  • Zdeněk Vejdělek and Miroslav Protiva
    N-substituted aminomethyl 4-cyclopentylphenyl ketones and 2-amino-1-(4-cyclopentylphenyl)ethanol: Synthesis and pharmacological screening
    1983, Vol. 48, Issue 2, pp. 642–648 [Abstract]
  • Zdeněk Polívka, Miroslav Rajšner, Jan Metyš, Jiří Holubek, Emil Svátek, Miroslav Ryska and Miroslav Protiva
    Antiaminic agents derived from thieno[2,3-c]-2-benzothiepin: 4-(1-Methyl-4-piperidylidene)-4,9-dihydrothieno[2,3-c]-2-benzothiepin and some related compounds
    1983, Vol. 48, Issue 2, pp. 623–641 [Abstract]
  • Jiří Křepelka, Drahuše Vlčková, Jiří Holubek and Jiří Roubík
    8-Substitution derivatives of D-6-methylergoline-I
    1983, Vol. 48, Issue 1, pp. 312–318 [Abstract]
  • Jiří Křepelka, Jan Beneš, Vladimír Pouzar, Jaroslav Vachek and Jiří Holubek
    Some 2-substitution derivatives of 5-(4-oxo-6-hydroxy-3,4-dihydro-5-pyrimidinyl)pentanoic acid
    1983, Vol. 48, Issue 1, pp. 304–311 [Abstract]
  • Miroslav Rajšner, Jan Metyš, Jiří Holubek and Miroslav Protiva
    Potential antidepressants: Some N-substituted derivatives of (E)-11-(3-methylaminopropylidene)-6,11-dihydrodibenzo[b,e]thiepin
    1983, Vol. 48, Issue 1, pp. 163–172 [Abstract]
  • Zdeněk Vejdělek, Marie Bartošová and Miroslav Protiva
    N-(Aminoacyl) and N-(aminoalkyl) derivatives of 4-cyclopentylaniline and N-ethyl-4-cyclopentylaniline; Synthesis and pharmacological screening
    1983, Vol. 48, Issue 1, pp. 156–162 [Abstract]
  • Karel Šindelář, Jiřina Metyšová, Jiří Holubek, Emil Svátek, Miroslav Ryska and Miroslav Protiva
    Fluorinated tricyclic neuroleptics with prolonged action: 3-Fluoro-10-[4-(2-hydroxyethyl)piperazino]-10,11-dihydrodibenzo[b,f]thiepins with less common substituents in position 8
    1983, Vol. 48, Issue 1, pp. 144–155 [Abstract]
  • Zdeněk J. Vejdělek, Jan Metyš and Miroslav Protiva
    S-Substituted derivatives of 8-chloro-6-(2-chlorophenyl)-1-mercaptomethyl-4H-s-triazolo[4,3-a]-1,4-benzodiazepine; Synthesis and pharmacology
    1983, Vol. 48, Issue 1, pp. 123–136 [Abstract]
  • Zdeněk Vejdělek, Jiří Holubek, Marie Bartošová and Miroslav Protiva
    4-(Aminoacylamido)-s-hydrindacenes and related compounds: Synthesis and pharmacological screening
    1982, Vol. 47, Issue 12, pp. 3297–3305 [Abstract]
  • Miroslav Protiva, Zdeněk Šedivý, Jiří Holubek, Emil Svátek, Jiřina Metyšová and Marie Bartošová
    Potential psychotropic and antihistamine agents: 1- and 3-alkyl-9-(3-dimethylaminopropylidene)-thioxanthenes and 3-alkyl-11-piperazino-10,11-dihydrodibenzo[b,f]thiepins
    1982, Vol. 47, Issue 11, pp. 3134–3147 [Abstract]
  • Karel Šindelář, Jiří Holubek, Emil Svátek, Miroslav Ryska, Antonín Dlabač, Jiřina Metyšová and Miroslav Protiva
    Tricyclic psychotropic agents containing two chalcogen atoms in the central ring: 2-Fluoro-8-substituted 6-(4-piperidyl)-6H-dibenz[b,e]-1,4-oxathiepins
    1982, Vol. 47, Issue 11, pp. 3114–3133 [Abstract]
  • Miroslav Protiva, Karel Šindelář, Vladimír Valenta, Jiří Holubek, Emil Svátek, Miroslav Ryska, Jiří Schlanger, Jiří Urban and Marta Hrubantová
    Reactions of 11-chloro-11-phenyl-6,11-dihydrodibenzo[b,e]-thiepin with piperidine and some further nucleophiles
    1982, Vol. 47, Issue 11, pp. 3094–3113 [Abstract]
  • Karel Šindelář, Jiřina Metyšová, Jiří Holubek, Emil Svátek, Jiří Protiva and Miroslav Protiva
    Tricyclic psychotropic agents containing two chalcogen atoms in the central ring: 8-Substituted 6-(4-piperidyl)-6H-dibenz[b,e]-1,4-oxathiepins
    1982, Vol. 47, Issue 11, pp. 3077–3093 [Abstract]
  • Miroslav Holub, Zdeněk Samek, Miloš Buděšínský, David Šaman, Ełżbieta Błoszyk and Bohdan Drożdż
    8α-Hydroxybalchanin - A new sesquiterpenic lactone from Leucanthemella serotina (L.) TZVEL.
    1982, Vol. 47, Issue 11, pp. 2927–2931 [Abstract]
  • Patricia Sierra, Ladislav Novotný, Zdeněk Samek, Miloš Buděšínský, Ladislav Dolejš and Karel Bláha
    Alkaloids of Rauvolfia salicifolia GRISEB species
    1982, Vol. 47, Issue 11, pp. 2912–2921 [Abstract]
  • Miloš Buděšínský, David Šaman and Zdeněk Wimmer
    Conformation studies of isomeric 1-acyloxy-2-(4-methoxybenzyl)-cyclohexanes by 1H NMR spectroscopy
    1982, Vol. 47, Issue 10, pp. 2763–2767 [Abstract]
  • Josef Hájíček, Jiří Holubek and Jan Trojánek
    Synthesis of 4,4- and 5,5-disubstituted 4,5-dihydro-6H-canthin-6-ones
    1982, Vol. 47, Issue 10, pp. 2749–2762 [Abstract]
  • Miroslav Kuchař, Václav Rejholec, Bohumila Brunová, Jaroslava Grimová, Oluše Matoušová, Oldřich Němeček and Hana Čepeláková
    Benzyloxyarylaliphatic acids: Synthesis and quantitative relations between structure and antiinflammatory activity
    1982, Vol. 47, Issue 9, pp. 2514–2524 [Abstract]
  • Zdenko Procházka, Miloš Buděšínský, Jorga Smolíková, Petr Trška and Karel Jošt
    1-Aminocyclopropanecarboxylic acid and its derivatives
    1982, Vol. 47, Issue 8, pp. 2291–2305 [Abstract]
  • Zdeněk Buděšínský, František Šmejkal and Miloš Buděšínský
    Some 1-β-D-ribofuranosyl-5-phenylcytosines and -5-(2-chlorophenyl)-2-thiocytosine
    1982, Vol. 47, Issue 8, pp. 2145–2149 [Abstract]
  • Ivan Beneš, Tomáš Vaněk and Miloš Buděšínský
    Nardiin, a new ent-kaurane diterpenoid from the liverwort Nardia scalaris
    1982, Vol. 47, Issue 7, pp. 1873–1877 [Abstract]
  • Jiří Křepelka, Iva Vančurová, Jiří Holubek, Milan Mělka and Karel Řežábek
    Derivatives of benzo(c)fluorene: II. Synthesis and biological effect of basic ethers of 7-oxo-7H-benzo(c)fluorene
    1982, Vol. 47, Issue 7, pp. 1856–1866 [Abstract]
  • Jan Beneš and Jiří Holubek
    1,2-Fused derivatives of ergoline
    1982, Vol. 47, Issue 6, pp. 1641–1644 [Abstract]
  • Jan Beneš and Jiří Holubek
    Wittig type reactions of 2-formylated derivatives of 6-methylergoline - I
    1982, Vol. 47, Issue 6, pp. 1636–1640 [Abstract]
  • Jiří Jílek, Josef Pomykáček, Jiřina Metyšová and Miroslav Protiva
    Fluorinated tricyclic neuroleptics with prolonged action: 8-Methoxy, 8-ethoxy, 8-ethylthio and 8-hydroxy derivatives of 3-fluoro-10-(4-methylpiperazino)-10,11-dihydrodibenzo[b,f]thiepin
    1982, Vol. 47, Issue 5, pp. 1382–1391 [Abstract]
  • Karel Šindelář, Jiří Holubek, Emil Svátek, Miroslav Ryska, Antonín Dlabač and Miroslav Protiva
    Tricyclic psychotropic agents containing two chalcogen atoms in the central ring: Synthesis of 6-(aminoalkyl) derivatives of 6H-dibenz[b,e]-1,4-oxathiepin
    1982, Vol. 47, Issue 5, pp. 1367–1381 [Abstract]
  • Jiří Křepelka, Jiří Roubík, Jiří Holubek and Iva Vančurová
    5-, 6- And 7-substitution derivatives of 7-oxo-7H-benzo(c)fluorene
    1982, Vol. 47, Issue 4, pp. 1258–1266 [Abstract]
  • Jiří Křepelka, Iva Vančurová and Jiří Holubek
    Reactions of 4-aryl-1-methoxynaphtalene-2,3-dicarboxylic acid anhydrides and naphtho(2,3-c)furan-1-(3H)-one derivatives with hydrazines
    1982, Vol. 47, Issue 4, pp. 1252–1257 [Abstract]
  • Karel Bláha, Miloš Buděšínský, Zdena Koblicová, Petr Maloň, Miloš Tichý, J. R. Baker, M. B. Hossain and Dick Van der Helm
    Optically active tricyclic dilactams with non-planar cis-amide groups: Synthesis, X-ray, NMR and CD studies
    1982, Vol. 47, Issue 3, pp. 1000–1019 [Abstract]
  • Vladimír Valenta, Jan Metyš and Miroslav Protiva
    (6,11-Dihydrodibenzo[b,e]thiepin-11-yl)methylamine, (4-methoxy-6,11-dihydrodibenzo[b,e]thiepin-11-yl)-methylamine and derivatives; Synthesis and pharmacological screening
    1982, Vol. 47, Issue 3, pp. 984–993 [Abstract]
  • Karel Šindelář, Jiří Holubek, Miroslav Ryska, Antonín Dlabač, Jiřina Metyšová, Emil Svátek, Marta Hrubantová, Jiří Protiva and Miroslav Protiva
    Tricyclic psychotropic agents containing two chalcogen atoms in the central ring: Derivatives of 11H-dibenz[b,f]-1,4-oxathiepin
    1982, Vol. 47, Issue 3, pp. 967–983 [Abstract]
  • Miroslav Holub, Miloš Buděšínský, Zdeněk Samek, Bohdan Drożdż, Halina Grabarczyk, Ayhan Ulubelen, Sevil Öksüz and Urszula Rychłewska
    Absolute configuration of xerantholide, a sesquiterpenic lactone from Anthemis austriaca JACQ.
    1982, Vol. 47, Issue 2, pp. 670–675 [Abstract]
  • Josef Jizba, Miloš Buděšínský, Tomáš Vaněk, A. Boeva, Kalinka Dimitrova, František Šantavý and Ladislav Novotný
    Components of Senecio pancicii DEGEN var. arnautorum (VELEN.) STOJ., STEF. et KIT. and S. Pancicii DEGEN var. pancicii
    1982, Vol. 47, Issue 2, pp. 664–669 [Abstract]
  • Juraj Harmatha, Miloš Buděšínský and Antonín Trka
    The structure of yatein. Determination of the positions, and configurations of benzyl groups in lignans of the 2,3-dibenzylbutyrolactone type
    1982, Vol. 47, Issue 2, pp. 644–663 [Abstract]
  • Miroslav Protiva, Zdeňka Kopicová and Jaroslava Grimová
    Synthesis of several 1-(aminoacyl)-4-cinnamylpiperazines as potential analgetics
    1982, Vol. 47, Issue 2, pp. 636–643 [Abstract]
  • Jiří Křepelka, Iva Vančurová, Jiří Holubek, Jiří Roubík and Drahuše Vlčková
    Syntheses and antineoplastic effects of some N-substituted imides of 1-substituted 4-aryl-naphthalene-2,3-dicarboxylic acids
    1982, Vol. 47, Issue 1, pp. 304–314 [Abstract]
  • Karel Šindelář, Jiří Holubek, Miroslav Ryska, Emil Svátek, Antonín Dlabač, Marta Hrubantová and Miroslav Protiva
    Tricyclic psychotropic agents containing two chalcogen atoms in the central ring: Synthesis of 11-(dimethylaminoalkyl) derivatives of 11H-dibenzo[b,e]-1,4-dioxepin and 11H-dibenzo[b,e]-1,4-dithiepin
    1982, Vol. 47, Issue 1, pp. 72–87 [Abstract]
  • Miroslav Rajšner, Emil Svátek, Jan Metyš and Miroslav Protiva
    Antidepressant fluorinated prothiadene derivatives: 9-Fluoro and 2,9-difluoro derivative of 11-(3-dimethylaminopropylidene)-6,11-dihydrodibenzo[b,e]thiepin
    1982, Vol. 47, Issue 1, pp. 65–71 [Abstract]
  • Bohumír Koutek, Libuše Pavlíčková, Miloš Buděšínský and Milan Souček
    Synthesis and properties of benzoannelated 6-(1,3-dithiolan-2-yliden)-2,4-cyclohexadien-1-ones
    1982, Vol. 47, Issue 1, pp. 59–64 [Abstract]
  • Jiří Jílek, Josef Pomykáček, Jiří Němec and Miroslav Protiva
    1-(3-Dimethylamino-1-phenylpropyl)piperazines and related compounds: Synthesis and pharmacological screening
    1981, Vol. 46, Issue 11, pp. 2729–2733 [Abstract]
  • Zdeněk Buděšínský, Miloš Buděšínský and Alois Šváb
    Addition of 2-methylthio-5-pyrimidinol and 5-methoxy-2-pyrimidinethiol to the acetylene triple bond
    1981, Vol. 46, Issue 9, pp. 2254–2262 [Abstract]
  • Miroslav Protiva, Zdeněk Šedivý, Josef Pomykáček, Václav Bártl, Jiří Holubek and Emil Svátek
    Potential metabolites of the noncataleptic neuroleptics: Synthesis of 2-chloro-6-hydroxy(and methoxy)-10-[4-(2-hydroxyethyl)piperazino]-10,11-dihydrodibenzo[b,f]thiepin
    1981, Vol. 46, Issue 9, pp. 2245–2253 [Abstract]
  • Zdeněk Vejdělek, Jiří Holubek, Marie Bartošová and Miroslav Protiva
    1-(4-Cyclopentylphenyl)ethylamine and derivatives: Synthesis and pharmacological screening
    1981, Vol. 46, Issue 9, pp. 2234–2244 [Abstract]
  • Zdeněk Polívka, Jiří Holubek, Emil Svátek, Jiřina Metyšová and Miroslav Protiva
    Fluorinated tricyclic neuroleptics: Synthesis and pharmacology of 2-chloro-8-fluoro-4-(4-methylpiperazino)-4,5-dihydrothieno[2,3-b]-1-benzothiepin
    1981, Vol. 46, Issue 9, pp. 2222–2233 [Abstract]
  • Jiří Křepelka, Iva Vančurová, Jiří Holubek and Jiří Roubík
    Hydrolytic products of 4-aryl-2,3-dicyano-1-naphthol derivatives
    1981, Vol. 46, Issue 9, pp. 2207–2216 [Abstract]
  • Jiří Křepelka and Jiří Holubek
    The synthesis of model lactones of cyclolignan type
    1981, Vol. 46, Issue 9, pp. 2123–2128 [Abstract]
  • Jiří Křepelka, Jiří Roubík and Jiří Holubek
    1-Substitution derivatives of 4-aryl-2,3-dibromo-1-naphthol
    1981, Vol. 46, Issue 9, pp. 2116–2122 [Abstract]
  • Miroslav Protiva, Karel Šindelář, Zdeněk Šedivý, Jiří Holubek and Marie Bartošová
    Potential metabolites of tricyclic neuroleptics: 3,7-Dimethoxy and 7,8-dimethoxy derivatives of 10-(4-methylpiperazino)-10,11-dihydrodibenzo[b,f]thiepin
    1981, Vol. 46, Issue 8, pp. 1808–1817 [Abstract]
  • Zdeněk Vejdělek, Marie Bartošová and Miroslav Protiva
    3-(s-Hydrindacen-4-yl)propylamines and 4-(s-hydrindacen-4-yl)butylamines; Synthesis and pharmacological screening
    1981, Vol. 46, Issue 8, pp. 1800–1807 [Abstract]
  • Miroslav Protiva, Karel Šindelář, Jiřina Metyšová, Jiří Holubek, Miroslav Ryska, Emil Svátek, Zdeněk Šedivý and Josef Pomykáček
    Fluorinated tricyclic neuroleptics with prolonged action: 3-Fluoro-8-halogeno derivatives of 10-piperazino-10,11-dihydrodibenzo[b,f]thiepins
    1981, Vol. 46, Issue 8, pp. 1788–1799 [Abstract]
  • Jiří Jílek, Josef Pomykáček, Jiřina Metyšová and Miroslav Protiva
    Neuroleptic agents derived from perathiepin: 6,7-Dichloro derivative of 10-(4-methylpiperazino)-10,11-dihydrodibenzo[b,f]thiepin and related compounds
    1981, Vol. 46, Issue 7, pp. 1607–1613 [Abstract]
  • Miroslav Rajšner, Antonín Dlabač and Miroslav Protiva
    Esters of 1-[4,4-bis(4-fluorophenyl)butyl]-4-(4-chloro-3-trifluoromethylphenyl)-4-piperidinol
    1981, Vol. 46, Issue 6, pp. 1530–1533 [Abstract]
  • Jiří Křepelka, Iva Vančurová and Jiří Holubek
    Some derivatives of 4-aryl-2,3-dicyano-1-naphthol
    1981, Vol. 46, Issue 6, pp. 1523–1529 [Abstract]
  • Vladimír Valenta, Marie Bartošová and Miroslav Protiva
    1-[3-(2-Alkoxyphenoxy)-3-phenylpropyl]piperazines and some related compounds
    1981, Vol. 46, Issue 5, pp. 1280–1287 [Abstract]
  • Miroslav Protiva, Zdeněk Šedivý, Josef Pomykáček, Emil Svátek and Jiří Holubek
    Potential metabolites of the neuroleptic agent octoclothepin; Synthesis of 8-chloro-2,6-dihydroxy and 8-chloro-3,6-dihydroxy derivatives of 10-(4-methylpiperazino)-10,11-dihydrodibenzo[b,f]thiepin
    1981, Vol. 46, Issue 5, pp. 1199–1209 [Abstract]
  • Irena Červená, Marta Hrubantová, Marie Bartošová and Miroslav Protiva
    Synthesis of arylthioacetamidoximes as potential antidepressants
    1981, Vol. 46, Issue 5, pp. 1188–1198 [Abstract]
  • Vladimír Valenta, Antonín Dlabač and Miroslav Protiva
    Potential noncataleptic neuroleptic agents: 2,4-Dichloro- and 2,4,8-trichloro-10-piperazino-10,11-dihydrodibenzo[b,f]thiepins
    1981, Vol. 46, Issue 3, pp. 781–791 [Abstract]
  • Ladislav Kniežo, Pavol Kristian, Miloš Buděšínský and Katarína Havrilová
    Stereochemical course of the reaction of 2-haloethyl isothiocyanates with nucleophiles. Stereospecific route to 4,5-disubstituted Δ2-thiazolines and thiazolidine-2-thiones
    1981, Vol. 46, Issue 3, pp. 717–728 [Abstract]
  • Karel Šindelář, Jiří Holubek, Jan Metyš, Marie Bartošová and Miroslav Protiva
    Synthesis of 3-(2-alkoxyphenoxy)-2-methyl (or phenyl)propylamines as potential antidepressants
    1981, Vol. 46, Issue 3, pp. 597–606 [Abstract]
  • Zdeněk Vejdělek, Emil Svátek, Jiří Holubek, Jan Metyš, Marie Bartošová and Miroslav Protiva
    Synthesis and pharmacological screening of 1-[2-tert-aminoethyl]-8-fluoro-5-[4-fluorophenyl]-2,3,4,5-tetrahydro-1H-1-benzazepines, their 1-[aminoacetyl] analogues and 1-substituted 9-fluoro-6-[4-fluorophenyl]-5,6-dihydro-4H-s-triazolo[4,3-a]-1-benzazepines
    1981, Vol. 46, Issue 1, pp. 148–160 [Abstract]
  • Václav Bártl, Jiřina Metyšová and Miroslav Protiva
    2-Chloro-7-fluoro- and 2-chloro-3,7-difluoro-11-[4-(4-fluoroaralkyl)piperazino]-10,11-dihydrodibenzo-[b,f]thiepins and related compounds; Long acting tranquillizers
    1981, Vol. 46, Issue 1, pp. 141–147 [Abstract]
  • Karel Šindelář, Miroslav Ryska, Jiří Holubek, Emil Svátek, Jiřina Metyšová, Jiří Protiva and Miroslav Protiva
    Fluorinated tricyclic neuroleptics with prolonged action: 3-Fluoro-8-trifluoromethyl derivatives of 10-(4-methylpiperazino)- and 10-[4-(2-hydroxyethyl)piperazino]-10,11-dihydrodibenzo-[b,f]thiepin
    1981, Vol. 46, Issue 1, pp. 118–140 [Abstract]
  • Zdeněk Vejdělek, Miroslav Rajšner, Antonín Dlabač, Miroslav Ryska, Jiří Holubek, Emil Svátek and Miroslav Protiva
    Psychotropic derivatives of 5-phenyl-7-chloro-1,3-dihydro-1,4-benzodiazepin-2-one and contribution to the synthesis of its 5-(2-chlorophenyl) analogue
    1980, Vol. 45, Issue 12, pp. 3593–3615 [Abstract]
  • Miroslav Semonský, Antonín Černý, Jiří Křepelka, Rudolf Kotva, Bohumil Kakáč, Jiří Holubek and Jaroslav Vachek
    Some ω-(2-amino-6-hydroxy-4-oxo-3,4-dihydro-5-pyrimidinyl) alkanoic acids, their derivatives and analogues
    1980, Vol. 45, Issue 12, pp. 3583–3592 [Abstract]
  • Václav Bártl, Antonín Dlabač and Miroslav Protiva
    Tricyclic potential neuroleptics: 2-chloro-11-[4-(4-fluoroaralkyl)piperazino]-10,11-dihydrodibenzo[b,f]thiepins and related compounds
    1980, Vol. 45, Issue 11, pp. 3182–3189 [Abstract]
  • Karel Šindelář, Jiří Jílek, Jiří Körbl, Fedir Jančik, Emil Svátek, Jiřina Metyšová and Miroslav Protiva
    Potential metabolites of the neuroleptic agent chlorprothixene; synthesis and pharmacology of the 3-, 4-, 6- and 7-hydroxy and methoxy derivatives of 2-chloro-9-(3-dimethylaminopropylidene)-thioxanthenes
    1980, Vol. 45, Issue 11, pp. 3166–3181 [Abstract]
  • Miloš Buděšínský, Zdeněk Samek and Miloš Tichý
    In situ reactions of amines and amino alcohols and their application to structural assignment by 1H NMR spectroscopy
    1980, Vol. 45, Issue 10, pp. 2784–2803 [Abstract]
  • Jiří Křepelka, Viktor Zikán, Jiří Holubek and Miroslav Semonský
    Derivatives of 4-aryl-2,3-dihalogeno-1-naphthol
    1980, Vol. 45, Issue 10, pp. 2700–2705 [Abstract]
  • Jiří Křepelka, Jiří Holubek and Miroslav Semonský
    Esters of 4,4-bis(4-ethylphenyl)-2,3-dibromo-2-butenoic acid and 7-ethyl-4-(4-ethylphenyl)-2,3-dibromo-1-naphthol
    1980, Vol. 45, Issue 10, pp. 2695–2699 [Abstract]
  • Irena Červená, Marta Hrubantová, Emil Svátek, Jiří Holubek, Miroslav Ryska, Jiřina Metyšová and Miroslav Protiva
    Fluorinated analogues of tricyclic neuroleptics: 6,9-difluoro derivative of 10-(4-methylpiperazino)-10,11-dihydrodibenzo[b,f]thiepin
    1980, Vol. 45, Issue 10, pp. 2688–2694 [Abstract]
  • Karel Šindelář, Emil Svátek, Jiří Holubek, Miroslav Ryska, Jiřina Metyšová, Zdeněk Šedivý and Miroslav Protiva
    Fluorinated analogues of the tricyclic neuroleptics; 7-Fluoro and 7-trifluoromethyl derivative of 10-(4-methylpiperazino)-10,11-dihydrodibenzo[b,f]thiepin
    1980, Vol. 45, Issue 4, pp. 1086–1098 [Abstract]
  • Jiří Křepelka, Jiří Holubek and Miroslav Semonský
    Some condensation products of ergoline - I Derivatives with ketones
    1980, Vol. 45, Issue 3, pp. 755–760 [Abstract]
  • Zdeněk Buděšínský, Josef Vavřina, Leon Langšádl and Jiří Holubek
    On the synthesis of 4- and 5-pyrimidinyl-diphenyl-(1-imidazolyl)methanes and their antifungal activity
    1980, Vol. 45, Issue 2, pp. 539–547 [Abstract]
  • Vladimír Valenta, Antonín Dlabač, Marie Bartošová, Emil Svátek and Miroslav Protiva
    10-[4-(3-Hydroxypropyl)piperazino]-8-methylsulfonyl-10,11-dihydrodibenzo[b,f]thiepin and some related potential metabolites of the neuroleptic agents oxyprothepin and methiothepin
    1980, Vol. 45, Issue 2, pp. 529–538 [Abstract]
  • Vladimír Valenta, Marie Bartošová and Miroslav Protiva
    Carbamates and ureas derived from 11-amino-6,11-dihydrodibenzo[b,e]thiepin; Synthesis and pharmacological screening
    1980, Vol. 45, Issue 2, pp. 517–528 [Abstract]
  • Jiří Jílek, Josef Pomykáček, Antonín Dlabač, Marie Bartošová and Miroslav Protiva
    Neuroleptics of the 8-methylthio-10-piperazino-10,11-dihydrodibenzo[b,f]thiepin series: New compounds and new procedures
    1980, Vol. 45, Issue 2, pp. 504–516 [Abstract]
  • Karel Šindelář, Jiří Holubek, Emil Svátek and Miroslav Protiva
    Synthesis of 3-chloro-5-(4-methylpiperazino)-6,7-dihydro-5H-dibenzo[b,g]thiocin, an eight-membered ring homologue of the neuroleptic agent octoclothepin
    1980, Vol. 45, Issue 2, pp. 491–503 [Abstract]
  • Karel Šindelář, Jiří Holubek, Emil Svátek, Miroslav Ryska, Jiřina Metyšová, Zdeněk Šedivý and Miroslav Protiva
    Potential metabolites of the neuroleptic agents noroxyclothepin and oxyclothepin; Synthesis of 8-chloro-3-hydroxy-10-[4-(2-hydroxyethyl)piperazino]- and -10-[4-(3-hydroxypropyl)piperazino]-10,11-dihydrodibenzo[b,f]thiepin
    1979, Vol. 44, Issue 12, pp. 3617–3626 [Abstract]
  • Zdeněk Vejdělek, Miroslav Rajšner, Emil Svátek, Jiří Holubek and Miroslav Protiva
    Synthesis of 7-chloro-5-(6,7,8,9-tetrahydro-5H-benzocyclohepten-2-yl)-2-methylamino-3H-1,4-benzodiazepine 4-oxide and of some related compounds
    1979, Vol. 44, Issue 12, pp. 3604–3616 [Abstract]
  • Vladimír Valenta, Emil Svátek, Antonín Dlabač, Marie Bartošová and Miroslav Protiva
    Noncataleptic neuroleptics: Potential metabolites of 2-chloro-10-[4-(2-hydroxyethyl)piperazino]-10,11-dihydrodibenzo[b,fthiepin
    1979, Vol. 44, Issue 10, pp. 3008–3018 [Abstract]
  • Miroslav Rajšner, František Mikšík, Jiřina Metyšová and Miroslav Protiva
    Fluorinated tricyclic neuroleptics: Synthesis and pharmacology of 8-fluoro-4-(4-methylpiperazino)-4,5-dihydrothieno[2,3-b]-1-benzothiepin
    1979, Vol. 44, Issue 10, pp. 2997–3007 [Abstract]
  • Miroslav Protiva, Karel Šindelář, Zdeněk Šedivý and Josef Pomykáček
    Potential metabolites of tricyclic neuroleptics: 2,8-Dihydroxy and 3,8-dihydroxy derivatives of 10-(4-methylpiperazino)-10,11-dihydrodibenzo[b,f]thiepin
    1979, Vol. 44, Issue 10, pp. 2987–2996 [Abstract]
  • Vladimír Valenta, František Kvis, Jiří Němec and Miroslav Protiva
    6,11-Dihydrodibenzo[b,e]thiepin-11-thiol and 11-acetic acid derivatives; Some 2-methyl-6,11-dihydrodibenzo[b,e]thiepins; Synthesis and pharmacological screening
    1979, Vol. 44, Issue 9, pp. 2689–2701 [Abstract]
  • Vladimír Valenta, Jiří Jílek, Josef Pomykáček, Antonín Dlabač, Martin Valchář, Jan Metyš and Miroslav Protiva
    Noncataleptic potential neuroleptics: 2-Methyl-10-(4-methylpiperazino)- and -10-[4-(2-hydroxyethyl)piperazino]-10,11-dihydrodibenzo[b,f]thiepin
    1979, Vol. 44, Issue 9, pp. 2677–2688 [Abstract]
  • Miroslav Rajšner, Václav Bártl, Karel Šindelář, Emil Svátek, Jiří Holubek, Jan Metyš and Miroslav Protiva
    Synthesis of new dibenzo[b,e]thiepin derivatives related to the antidepressant agent prothiadene
    1979, Vol. 44, Issue 8, pp. 2536–2549 [Abstract]
  • Irena Červená, Jiřina Metyšová, Václav Bártl and Miroslav Protiva
    Fluorinated neuroleptics of the 10-piperazino-10,11-dihydrodibenzo[b,f]thiepin series; 6-Fluoro derivatives of perathiepin, octoclothepin, doclothepin and some related compounds
    1979, Vol. 44, Issue 7, pp. 2139–2155 [Abstract]
  • Jiří O. Jílek, Jiří Holubek, Emil Svátek, Miroslav Ryska, Josef Pomykáček and Miroslav Protiva
    Reaction of some 3-(phenylthioaryl)propionic acids with polyphosphoric acid; Formation of 2H-cyclopenta[k,l]thioxanthenes
    1979, Vol. 44, Issue 7, pp. 2124–2138 [Abstract]
  • Miroslav Protiva, Karel Šindelář, Zdeněk Šedivý and Jiřina Metyšová
    Potential metabolites of tricyclic neuroleptics and their fluorinated analogues; 3-Hydroxy-, 3-methoxy- and 3-fluoro-10-(4-methylpiperazino)-10,11-dihydrodibenzo[b,f]thiepin
    1979, Vol. 44, Issue 7, pp. 2108–2123 [Abstract]
  • Miloš Buděšínský, Miloslav Černý, Tomáš Trnka and Soňa Vašíčková
    1H NMR spectra and the conformation of 1,6 : 2,3- and 1,6 : 3,4-dianhydro-β-D-hexopyranoses and their derivatives
    1979, Vol. 44, Issue 6, pp. 1965–1983 [Abstract]
  • Miloš Buděšínský, Tomáš Trnka and Miloslav Černý
    The 1H NMR spectra and the conformation of 1,6-anhydro-β-D-hexopyranoses and their triacetates
    1979, Vol. 44, Issue 6, pp. 1949–1964 [Abstract]
  • Emil Svátek, Viktor Zikán and Miroslav Semonský
    Spectral manifestations of strong hydrogen bonds in seven-membered rings of pyrazolecarboxylic acid derivatives
    1979, Vol. 44, Issue 3, pp. 781–787 [Abstract]
  • Zdeněk Samek and Miloš Buděšínský
    In situ reactions with trichloroacetyl isocyanate and their application to structural assignment of hydroxy compounds by 1H NMR spectroscopy. A general comment
    1979, Vol. 44, Issue 2, pp. 558–588 [Abstract]
  • Jiří Klinot, Jarmil Světlý, Dagmar Kudláčková, Miloš Buděšínský and Alois Vystrčil
    Preparation of 2-methyl-3-oxo triterpenoids of 18α-oleanane series and the conformation of ring A
    1979, Vol. 44, Issue 1, pp. 211–225 [Abstract]
  • Jiří Jílek, Jiří Holubek, Emil Svátek, Marie Bartošová, Jiřina Metyšová, Josef Pomykáček and Miroslav Protiva
    8-Chloro-3-hydroxy-10-piperazino-10,11-dihydrodibenzo[b,f]thiepins, their O-methyl derivatives and further potential metabolites of the neuroleptic agent octoclothepin
    1978, Vol. 43, Issue 11, pp. 3092–3102 [Abstract]
  • Miroslav Protiva, Irena Červená, Miroslav Rajšner, Jiřina Metyšová and Marta Hrubantová
    Fluorinated tricyclic neuroleptics: 3-Fluoro and 3,6-difluoro derivatives of chlorprothixene and 6-fluoro-2-isopropyl derivative of prothixene
    1978, Vol. 43, Issue 10, pp. 2656–2663 [Abstract]
  • Jan Vrkoč, Miloš Buděšínský and Petr Sedmera
    Structure of 2α,3α-dihydroxy- and 2α,3β-dihydroxy-1(15),8(19)-trinervitadines from Nasututermes costalis (HOLMGREN)
    1978, Vol. 43, Issue 9, pp. 2478–2485 [Abstract]
  • Václav Bártl, Jiří Holubek, Jiří Němec, Marie Bartošová and Miroslav Protiva
    Derivatives of 8-chloro-10,11-dihydrodibenzo[b,f]thiepin-10-amine, -10-ol and -10-thiol; Synthesis and pharmacological screening
    1978, Vol. 43, Issue 9, pp. 2427–2443 [Abstract]
  • Huynh Kim Thoa, Želimír Procházka, Miloš Buděšínský and Pavel Kočovský
    Hydroxylation of 6β-methoxy-3α,5-cyclo-5α-androstan-17-one with Rhizopus nigricans
    1978, Vol. 43, Issue 9, pp. 2305–2311 [Abstract]
  • Jan Kovář, Ladislav Skurský and Miroslav Protiva
    Structural factors affecting interactions of tricyclic psychotropic drugs with alcohol dehydrogenase
    1978, Vol. 43, Issue 8, pp. 2068–2081 [Abstract]
  • Miroslav Rajšner, Zdeňka Kopicová, Jiří Holubek, Emil Svátek, Jan Metyš, Marie Bartošová, František Mikšík and Miroslav Protiva
    4,4-Bis(4-fluorophenyl)butylamines and their cyclic analogues; An efficient synthesis of the neuroleptic penfluridol
    1978, Vol. 43, Issue 7, pp. 1760–1777 [Abstract]
  • Jiří O. Jílek, Josef Pomykáček, Jiřina Metyšová, Marie Bartošová and Miroslav Protiva
    Potential metabolites of the neuroleptic agent octoclothepin; Synthesis and pharmacology of 8-chloro-6-hydroxy-10-(4-methylpiperazino)-10,11-dihydrodibenzo[b,f]thiepin and some related compounds
    1978, Vol. 43, Issue 7, pp. 1747–1759 [Abstract]
  • Zdeněk J. Vejdělek, Marie Bartošová, Miroslav Ryska and Miroslav Protiva
    2-(s-Hydrindacen-4-yl)ethylamines and their 1-methyl and 1,1-dimethyl derivatives; Synthesis and pharmacological screening
    1978, Vol. 43, Issue 7, pp. 1732–1746 [Abstract]
  • Viktor Zikán, Miroslav Semonský, Bohumil Kakáč, Jiří Holubek and Karel Řežábek
    Reactions of methyl esters of 3-bromo-4-(4-alkoxyphenyl)-4-oxo-2-butenoic acids with diethyl sodium malonate
    1978, Vol. 43, Issue 7, pp. 1727–1731 [Abstract]
  • Miroslav Rajšner, František Mikšík and Miroslav Protiva
    [5-Chloro-2-(phenylthio)phenyl]acetic acid, some derivatives and products of further transformations
    1978, Vol. 43, Issue 5, pp. 1276–1284 [Abstract]
  • Jan Vrkoč, Miloš Buděšínský and Petr Sedmera
    Structure of trinervitene diterpenoids from Nasutitermes rippertii (RAMBUR)
    1978, Vol. 43, Issue 4, pp. 1125–1133 [Abstract]
  • Zdeněk J. Vejdělek, Marie Bartošová, Alois Čapek and Miroslav Protiva
    4-(Aminoacetyl)-s-hydrindacenes and 2-amino-1-(s-hydrindacen-4-yl)-ethanols; Synthesis and pharmacological screening
    1978, Vol. 43, Issue 4, pp. 970–980 [Abstract]
  • Karel Šindelář, Jiří O. Jílek, Josef Pomykáček, Zdeněk Šedivý and Miroslav Protiva
    Synthesis of 2-acetyl and 3-acetyl derivatives of 8-chloro-10-(4-methylpiperazino)-10,11-dihydrodibenzo[b,f]-thiepin; 2-Acyl-7-substituted thioxanthenes
    1978, Vol. 43, Issue 2, pp. 471–497 [Abstract]
  • Huynh Kim Thoa, Václav Šašek, Miloš Buděšínský, Ivan Jablonský, Ludmila Eignerová, Nguyen Gia Chan and Želimír Procházka
    Biological transformation of 3β-hydroxy-5-androsten-17-one with the mushroom Pleurotus ostreatus (JACQ. ex FR.) KUMM.
    1978, Vol. 43, Issue 1, pp. 336–343 [Abstract]
  • Karel Šindelář, Antonín Dlabač and Miroslav Protiva
    Noncataleptic neuroleptics; 8-Chloro-2-hydroxy-11-(4-methylpiperazino)-5H-dibenzo[b,e]-1,4-diazepine as a potential metabolite of clozapine
    1978, Vol. 43, Issue 1, pp. 309–315 [Abstract]